Synthesis and in vitro protozoocidal evaluation of novel diazabicyclic tropolone derivatives

Archiv der Pharmazie

Volumn 340, Issue 11, 2007, Pages 569-576

  Khrizman, Alexander ^a   Slack, Rachel D ^a   Remsing, Richard C ^a   Little, Susan ^b   Yardley, Vanessa ^b   Moyna, Guillermo ^a  

^a UNIVERSITY OF THE SCIENCES   (United States)

^b LONDON SCHOOL OF HYGIENE AND TROPICAL MEDICINE   (United Kingdom)

Author keywords

Hydrazynes; Parasitoses; Protozoocidal activity; Synthesis; Tropolone derivatives

Indexed keywords

ANTIPARASITIC AGENT; TROPOLONE DERIVATIVE;

ARTICLE; DIELS ALDER REACTION; DRUG MECHANISM; EVALUATION; IN VITRO STUDY; LEISHMANIA DONOVANI; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; PROTOZOON; SYNTHESIS; TRYPANOSOMA CRUZI; TRYPANOSOMA RHODESIENSE;

ANIMALS; ANTIPROTOZOAL AGENTS; AZABICYCLO COMPOUNDS; CELL SURVIVAL; HUMANS; KB CELLS; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; PARASITIC SENSITIVITY TESTS; PROTOZOA; STRUCTURE-ACTIVITY RELATIONSHIP; TROPOLONE;

EID: 36549077336     PISSN: 03656233     EISSN: 15214184     Source Type: Journal    
DOI: 10.1002/ardp.200700143     Document Type: Article

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