Unique spirocyclopiperazinium salt III: Further investigation of monospirocyclopiperazinium (MSPZ) salts as potential analgesics

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 22, 2007, Pages 6245-6249

  Sun, Qi ^a   Yue, Cai Qin ^a   Ye, Jia ^a   Li, Chang Ling ^a   Cheng, Tie Ming ^a   Li, Run Tao ^a  

^a PEKING UNIVERSITY HEALTH SCIENCE CENTER   (China)

Author keywords

Analgesic; Monospirocyclopiperazinium salts; Structure activity relationship; Synthesis

Indexed keywords

ANALGESIC AGENT; PIPERAZINE DERIVATIVE; SPIROCYCLOPIPERAZINIUM DERIVATIVE; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANALGESICS; ANIMALS; DIMETHYLPHENYLPIPERAZINIUM IODIDE; DRUG EVALUATION, PRECLINICAL; MICE; MOLECULAR STRUCTURE; PAIN MEASUREMENT; PIPERAZINES; SALTS; SPIRO COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 35048845088     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.09.026     Document Type: Article

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