Methyl 2-(2-(4-formylphenoxy)acetamido)-2-substituted acetate derivatives: A new class of acetylcholinesterase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 8, 2007, Pages 2123-2125

  Wen, Huan ^a   Zhou, Yayao ^a   Lin, Chonglan ^a   Ge, Hui ^a   Ma, Lin ^a   Wang, Zihou ^b   Peng, Wenlie ^a   Song, Huacan ^a  

^a SUN YAT SEN UNIVERSITY   (China)

^b State Drug Administration   (China)

Author keywords

4 Hydroxybenzaldehyde; AChE inhibitors; Methyl 2 (2 (4 formylphenoxy) acetamido) 2 substituted acetate; Synthesis

Indexed keywords

ACETIC ACID DERIVATIVE; CHOLINESTERASE INHIBITOR; DONEPEZIL; GALANTAMINE; RIVASTIGMINE; TACRINE;

ARTICLE; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION;

ACETATES; ALZHEIMER DISEASE; BENZALDEHYDES; CHOLINESTERASE INHIBITORS; HUMANS; INHIBITORY CONCENTRATION 50; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33947608612     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.01.091     Document Type: Article

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