In vitro efficiency of new acridyl derivatives against Plasmodium falciparum

Bioorganic and Medicinal Chemistry

Volumn 15, Issue 9, 2007, Pages 3278-3289

  Guetzoyan, Lucie ^a   Ramiandrasoa, Florence ^a   Dorizon, Hélène ^a   Desprez, Christine ^a   Bridoux, Alexandre ^a   Rogier, Christophe ^b   Pradines, Bruno ^b   Perrée Fauvet, Martine ^a  

^a UNIVERSITÉ PARIS SUD   (France)

^b SERVICE DE SANTÉ DES ARMÉES   (France)

Author keywords

Aminoacridine; Antimalarial; Peptidic synthesis; Plasmodium falciparum

Indexed keywords

1 [2 [8 (ACRIDIN 9 YLAMINO) 8 OXOOCTYLAMINO] 2 OXOETHYLAMINO] 5 [AMINO(IMINIO)METHYLAMINO] 1 OXOPENOXOPENTAN 2 AMMONIUM; 9 (6 AMMONIOHEXYLAMINO) 6 CHLORO 2 METHOXYACRIDININE; 9 [6 (4 AMMONIOBUTANAMIDO)HEXYLAMINO] 6 CHLORO 2 METHOXYACRIDININE; ACRIDINE DERIVATIVE; CHLOROQUINE; UNCLASSIFIED DRUG;

ANTIBIOTIC RESISTANCE; ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG INHIBITION; DRUG SENSITIVITY; DRUG SYNTHESIS; IC 50; IN VITRO STUDY; MICROBIAL GROWTH; NONHUMAN; PLASMODIUM FALCIPARUM; SUBSTITUTION REACTION;

ACRIDINES; ANIMALS; ANTIMALARIALS; MOLECULAR STRUCTURE; PARASITIC SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

PLASMODIUM FALCIPARUM;

EID: 33947604335     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2007.02.022     Document Type: Article

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