Syntheses of F-18 labeled fluoroalkyltyrosine derivatives and their biological evaluation in rat bearing 9L tumor

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 1, 2007, Pages 200-204

  Moon, Byung Seok ^a,b   Lee, Tae Sup ^a   Lee, Kyo Chul ^a   An, Gwang Il ^a   Cheon, Gi Jeong ^a   Lim, Sang Moo ^a   Choi, Chang Woon ^a   Chi, Dae Yoon ^b   Chun, Kwon Soo ^a  

^a Korea Institute of Radiation and Medical Science   (South Korea)

^b Inha University   (South Korea)

Author keywords

Amino acids; Labeled tyrosine; O (2 18F Fluoroethyl) l tyrosine (l 18F FET); PET; Tumor imaging

Indexed keywords

2 (2 FLUOROETHYL)TYROSINE F 18; 3 (3 FLUOROPROPYL)TYROSINE F 18; ACETONITRILE; FLUORINE DERIVATIVE; O METHYL 3 (2 FLUOROETHYL)TYROSINE F 18; O METHYL 3 (3 FLUOROPROPYL)TYROSINE F 18; TYROSINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; DRUG ACCUMULATION; DRUG BLOOD LEVEL; DRUG BRAIN LEVEL; DRUG DISTRIBUTION; DRUG HYDROLYSIS; DRUG MUSCLE LEVEL; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TUMOR LEVEL; GLIOMA; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RAT;

ANIMALS; BRAIN NEOPLASMS; FLUORINE RADIOISOTOPES; GLIOMA; RADIOPHARMACEUTICALS; RATS; RATS, INBRED F344; TISSUE EMBEDDING; TYROSINE;

RATTUS;

EID: 33845769514     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.09.063     Document Type: Article

References (22)

1. In: Hubner K.F., Collmann J., Buonocore E., and Kabalka G.W. (Eds). Clinical positron emission tomography (1991), Mosby, St. Louis, MO 110
2. Tang G.H. Acta Pharm. Sin. 36 (2001) 470
3. Laverman P., Boerman O.C., Corstens F.H.M., and Oyen W.J. Eur. J. Nucl. Med. 29 (2002) 681
4. Langstrom B., Antoni G., Gullberg P., Halldin C., Malmborg P., Nagren K., Rimland A., and Svard H. J. Nucl. Med. 28 (1987) 1037
5. Inoue T., Tomiyoshi K., Higuichi T., Ahmed K., Sarwar M., Aoyagi K., Amano S., Alyafei S., Zhang H.N., and Endo K. J. Nucl. Med. 39 (1998) 663
6. Kubota K., Ishiwata K., Kubota R., Yamada S., Takahashi J., Abe Y., Fukuda H., and Ido T. J. Nucl. Med. 37 (1996) 320
7. Shoup T.M., Olson J., Hoffman J.M., Votaw J., Eshima D., Eshima L., Camp V.M., Stabin M., Votaw D., and Goodman M.M. J. Nucl. Med. 40 (1999) 331
8. Wester H.J., Herz M., Senekowitsch-Schmidtke R., Schwaiger M., Stocklin G., and Hamacher K. Nucl. Med. Biol. 26 (1999) 259
9. Bading J.R., Kan-Mitchell J., and Conti P.S. Nucl. Med. Biol. 23 (1996) 779
10. Ishiwata K., Ido T., Mejia A.A., Ichihashi M., and Mishima Y. Appl. Radiat. Isot. 42 (1991) 325
11. Langen K.J., Coenen H.H., Roosen N., Kling P., Muzik O., Herzog H., Kuwert T., Stocklin G., and Feinendegen L.E. J. Nucl. Med. 31 (1990) 281
12. Martarello L., McConathy J., Camp V.M., Malveaux E.J., Simpson N.E., Simpson C.P., Olson J.J., Bowers G.D., and Goodman M.M. J. Med. Chem. 45 (2002) 2250
13. Wester H.J., Herz M., Weber W., Heiss P., Senekowitsch-Schmidtke R., Schwaiger M., and Stocklin G. J. Nucl. Med. 40 (1999) 205
14. Heiss P., Mayer S., Herz M., Wester H.J., Schwaiger M., and Senekowitsch-Schmidtke R. J. Nucl. Med. 40 (1999) 1367
15. Tang G.H., Wang M.F., Tang X.L., Luo L., and Gan M.Q. Nucl. Med. Biol. 30 (2003) 733
16. Kaim A.H., Weber B., Kurrer M.O., Westera G., Schweitzer A., Gottschalk J., von Schulthess G.K., and Buck A. Eur. J. Nucl. Med. 29 (2002) 648
17. Rau F.C., Weber W.A., Wester H.J., Herz M., Becker I., Kruger A., Schwaiger M., and Senekowitsch-Schmidtke R. Eur. J. Nucl. Med. 29 (2002) 1039
18. Choe Y.S., Song D.H., Lee K.-J., Kim S.E., Choi Y., Lee K.H., Kim B.-T., Oh S.J., and Chi D.Y. Appl. Radiat. Isot. 49 (1998) 73
19. Barrio J.R., Petric A., Satyamurthy N., Huang S.C., and Yu D.C. J. Nucl. Med. 35S (1994) 83P
20. Lee K.C., Lee S.Y., Choe Y.S., and Chi D.Y. Bull. Korean Chem. Soc. 25 (2004) 1225
21. +) 256.1349. Found: 256.1349.
22. Moon B.S., Kim S.W., Lee T.S., Ahn S.H., Lee K.C., An G.I., Yang S.D., Chi D.Y., Choi C.W., Lim S.M., and Chun K.S. Bull. Korean Chem. Soc. 26 (2005) 91