-
1
-
-
0037139571
-
-
Janvier, P.; Sun, X.; Bienaymé, H.; Zhu, J. J. Am. Chem. Soc. 2002, 124, 2560-2567.
-
(2002)
J. Am. Chem. Soc.
, vol.124
, pp. 2560-2567
-
-
Janvier, P.1
Sun, X.2
Bienaymé, H.3
Zhu, J.4
-
2
-
-
0035903506
-
-
Wess, G.; Urmann, M.; Sickenberger, B. Angew. Chem., Int. Ed. 2001, 40, 3341-3350.
-
(2001)
Angew. Chem., Int. Ed.
, vol.40
, pp. 3341-3350
-
-
Wess, G.1
Urmann, M.2
Sickenberger, B.3
-
3
-
-
0024239320
-
-
Evans, B. E.; Rittle, K. E.; Bock, M. G.; DiPardo, R. M.; Freidinger, R. M.; Whitter, W. L.; Lundell, G. F.; Veber, D. F.; Anderson, P. S.; Chang, R. S. L.; Lotti, V. J.; Cerino, D. J.; Chen, T. B.; Kling, P. J.; Kunkel, K. A.; Springer, J. P.; Hirshfield, J. J. Med. Chem. 1988, 31, 2235-2246.
-
(1988)
J. Med. Chem.
, vol.31
, pp. 2235-2246
-
-
Evans, B.E.1
Rittle, K.E.2
Bock, M.G.3
Dipardo, R.M.4
Freidinger, R.M.5
Whitter, W.L.6
Lundell, G.F.7
Veber, D.F.8
Anderson, P.S.9
Chang, R.S.L.10
Lotti, V.J.11
Cerino, D.J.12
Chen, T.B.13
Kling, P.J.14
Kunkel, K.A.15
Springer, J.P.16
Hirshfield, J.17
-
4
-
-
0037529208
-
-
Lavilla, R.; Bernabeu, M. C.; Carranco, I.; Dias, J. L. Org. Lett. 2003, 5, 717-720.
-
(2003)
Org. Lett.
, vol.5
, pp. 717-720
-
-
Lavilla, R.1
Bernabeu, M.C.2
Carranco, I.3
Dias, J.L.4
-
5
-
-
33644947717
-
-
Evdokimov, N. M.; Magedov, I. V.; Kireev, A. S.; Kornienko, A. Org. Lett. 2006, 8, 899-902.
-
(2006)
Org. Lett.
, vol.8
, pp. 899-902
-
-
Evdokimov, N.M.1
Magedov, I.V.2
Kireev, A.S.3
Kornienko, A.4
-
6
-
-
0037060923
-
-
Doherty, G. A.; Kamenecka, T.; McCauley, E.; Van Riper, G.; Mumford, R. A.; Tong, S.; Hagmann, W. K. Bioorg. Med. Chem. Lett. 2002, 12, 729-731.
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 729-731
-
-
Doherty, G.A.1
Kamenecka, T.2
McCauley, E.3
Van Riper, G.4
Mumford, R.A.5
Tong, S.6
Hagmann, W.K.7
-
7
-
-
2542531589
-
-
Connolly, S.; Aberg, A.; Arvai, A.; Beaton, H. G.; Cheshire, D. R.; Cook, A. R.; Cooper, S.; Cox, D.; Hamley, P.; Mallinder, P.; Millichip, I.; Nicholls, D. J.; Rosenfeld, R. J.; St-Gallay, S. A.; Tainer, J.; Tinker, A. C.; Wallace, A. V. J. Med. Chem. 2004, 47, 3320-3323.
-
(2004)
J. Med. Chem.
, vol.47
, pp. 3320-3323
-
-
Connolly, S.1
Aberg, A.2
Arvai, A.3
Beaton, H.G.4
Cheshire, D.R.5
Cook, A.R.6
Cooper, S.7
Cox, D.8
Hamley, P.9
Mallinder, P.10
Millichip, I.11
Nicholls, D.J.12
Rosenfeld, R.J.13
St-Gallay, S.A.14
Tainer, J.15
Tinker, A.C.16
Wallace, A.V.17
-
8
-
-
33748947558
-
-
PCT Int Appl. WO 2005058315 A1 20050630, 2005
-
Chen, H.; Zhang, W.; Tam, R.; Raney, A. K. PCT Int Appl. WO 2005058315 A1 20050630, 2005.
-
-
-
Chen, H.1
Zhang, W.2
Tam, R.3
Raney, A.K.4
-
9
-
-
0034705043
-
-
Perrier, V.; Wallace, A. C.; Kanedo, K.; Safar, J.; Prusiner, S. B.; Cohen, F. E. Proc. Natl. Acad. Sci. U.S.A. 2000, 97, 6073-6078.
-
(2000)
Proc. Natl. Acad. Sci. U.S.A.
, vol.97
, pp. 6073-6078
-
-
Perrier, V.1
Wallace, A.C.2
Kanedo, K.3
Safar, J.4
Prusiner, S.B.5
Cohen, F.E.6
-
10
-
-
0035209620
-
-
Fredholm, B. B.; Ijzerman, A. P.; Jacobson, K. A.; Klotz, K.-N.; Linden, J. Pharmacol. Rev. 2001, 53, 527-552.
-
(2001)
Pharmacol. Rev.
, vol.53
, pp. 527-552
-
-
Fredholm, B.B.1
Ijzerman, A.P.2
Jacobson, K.A.3
Klotz, K.-N.4
Linden, J.5
-
12
-
-
29144448797
-
-
El Kaim, L.; Grimaud, L.; Oble, J. Angew. Chem., Int. Ed. 2005, 117, 7961-7964.
-
(2005)
Angew. Chem., Int. Ed.
, vol.117
, pp. 7961-7964
-
-
El Kaim, L.1
Grimaud, L.2
Oble, J.3
-
13
-
-
19944398117
-
-
Wang, H. Y.; Liao, Y. X.; Guo, Y. L.; Tang, Q. H.; Lu, L. Synlett 2005, 8, 1239-1242.
-
(2005)
Synlett
, vol.8
, pp. 1239-1242
-
-
Wang, H.Y.1
Liao, Y.X.2
Guo, Y.L.3
Tang, Q.H.4
Lu, L.5
-
14
-
-
10744219810
-
-
Cho, S. D.; Park, Y. D.; Kim, J. J.; Lee, S. G.; Ma, C.; Song, S. Y.; Joo, W. H.; Falck, J. R.; Shiro, M.; Shin, D. S.; Yoon, Y. J. J. Org. Chem. 2003, 68, 7918-7920.
-
(2003)
J. Org. Chem.
, vol.68
, pp. 7918-7920
-
-
Cho, S.D.1
Park, Y.D.2
Kim, J.J.3
Lee, S.G.4
Ma, C.5
Song, S.Y.6
Joo, W.H.7
Falck, J.R.8
Shiro, M.9
Shin, D.S.10
Yoon, Y.J.11
-
15
-
-
0001028934
-
-
Amino-6-trifluoro pyrimidines are reported to be potent therapeutic agents for malaria: Barlin, G. B.; Kotecka, B.; Rieckmann, K. H. Aust. J. Chem. 1996, 49, 647-650.
-
(1996)
Aust. J. Chem.
, vol.49
, pp. 647-650
-
-
Barlin, G.B.1
Kotecka, B.2
Rieckmann, K.H.3
-
16
-
-
0042320464
-
-
Sardarian, A.; Douglas, K. T.; Read, M.; Sims, P. F. G.; Hyde, J. E.; Chitnumsub, P.; Sirawaraporn, R.; Sirawaraporn, W. Org. Biomol. Chem. 2003, 1, 960-964.
-
(2003)
Org. Biomol. Chem.
, vol.1
, pp. 960-964
-
-
Sardarian, A.1
Douglas, K.T.2
Read, M.3
Sims, P.F.G.4
Hyde, J.E.5
Chitnumsub, P.6
Sirawaraporn, R.7
Sirawaraporn, W.8
-
19
-
-
84985097319
-
-
Burdeska, K.; Fuhrer, H.; Kabas, G.; Siegrist, A. E. Helv. Chim. Acta 1981, 64, 113-152.
-
(1981)
Helv. Chim. Acta
, vol.64
, pp. 113-152
-
-
Burdeska, K.1
Fuhrer, H.2
Kabas, G.3
Siegrist, A.E.4
-
20
-
-
0034597613
-
-
Norman, M. H.; Chen, N.; Chen, Z.; Fotsch, C.; Hale, C.; Han, N.; Hurt, R.; Jenkins, T.; Kincaid, J.; Liu, L.; Lu, Y.; Moreno, O.; Santora, V. J.; Sonnenberg, J. D.; Karbon, W. J. Med. Chem. 2000, 43, 4288-4312.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 4288-4312
-
-
Norman, M.H.1
Chen, N.2
Chen, Z.3
Fotsch, C.4
Hale, C.5
Han, N.6
Hurt, R.7
Jenkins, T.8
Kincaid, J.9
Liu, L.10
Lu, Y.11
Moreno, O.12
Santora, V.J.13
Sonnenberg, J.D.14
Karbon, W.15
-
21
-
-
84942709016
-
-
The rearrangement step observed in the Ugi processes was coined as Mumm rearrangement in relation to the imide-isoimide rearrangement studied by Mumm in 1910. Mumm, O. Ber. Dstch. Chem. Ges. 1910, 43, 886-893.
-
(1910)
Ber. Dstch. Chem. Ges.
, vol.43
, pp. 886-893
-
-
Mumm, O.1
-
22
-
-
0001521573
-
-
(a) Ugi, I.; Meyr, R.; Fetzer, U.; Steinbrückner, C. Angew. Chem. 1959, 71, 386.
-
(1959)
Angew. Chem.
, vol.71
, pp. 386
-
-
Ugi, I.1
Meyr, R.2
Fetzer, U.3
Steinbrückner, C.4
-
24
-
-
84982057469
-
-
(c) Ugi, I.; Rosendahl, F. K.; Bodesheim, F. Justus Liebigs Ann. Chem. 1963, 666, 54-61.
-
(1963)
Justus Liebigs Ann. Chem.
, vol.666
, pp. 54-61
-
-
Ugi, I.1
Rosendahl, F.K.2
Bodesheim, F.3
-
27
-
-
26844537872
-
-
For recent reviews concerning the Ugi coupling, see: (a) Banfi, L.; Riva, R. Org. React. 2005, 65, 1-140.
-
(2005)
Org. React.
, vol.65
, pp. 1-140
-
-
Banfi, L.1
Riva, R.2
-
29
-
-
1642338545
-
-
(c) Ugi, I.; Werner, B.; Dömling, A. Molecules 2003, 8, 53-66.
-
(2003)
Molecules
, vol.8
, pp. 53-66
-
-
Ugi, I.1
Werner, B.2
Dömling, A.3
-
31
-
-
0034665244
-
-
(e) Bienaymé, H.; Hulme, C.; Oddon, G.; Schmitt, P. Chem.-Eur. J. 2000, 6, 3321-3329.
-
(2000)
Chem.-Eur. J.
, vol.6
, pp. 3321-3329
-
-
Bienaymé, H.1
Hulme, C.2
Oddon, G.3
Schmitt, P.4
-
32
-
-
0001134412
-
-
(f) Dömling, A.; Ugi, I. Angew. Chem., Int. Ed. 2000, 39, 3168-3210.
-
(2000)
Angew. Chem., Int. Ed.
, vol.39
, pp. 3168-3210
-
-
Dömling, A.1
Ugi, I.2
|