Fatty acid synthase inhibitory activity of acylphloroglucinols isolated from Dryopteris crassirhizoma

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 18, 2006, Pages 4738-4742

  Na, MinKyun ^a   Jang, JunPil ^a   Min, Byung Sun ^b   Lee, Sang Jun ^c   Lee, Myung Sun ^a   Kim, Bo Yeon ^a   Oh, Won Keun ^a   Ahn, Jong Seog ^a  

^a Korea Research Institute of Bioscience and Biotechnology (KRIBB)   (South Korea)

^b Catholic University of Daegu   (South Korea)

^c AmorePacific Corporation   (South Korea)

Author keywords

Acylphloroglucinols; Dryopteridaceae; Dryopteris crassirhizoma; FAS inhibitors; Fatty acid synthase (FAS)

Indexed keywords

3 HYDROXYFLAVONE; ALBASPIDIN; ASPIDIN BB; ASPIDINOL; CERULENIN; EPICATECHIN; FATTY ACID SYNTHASE INHIBITOR; FILIXIC ACID; FLAVASPIDIC ACID; LUTEOLIN; METHYLENEBISMETHYLPHLOROBUTYROPHENONE; NORFLAVASPIDIC ACID; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; DRUG DETERMINATION; DRUG IDENTIFICATION; DRUG INHIBITION; DRUG ISOLATION; DRUG SCREENING; DRYOPTERIS; DRYOPTERIS CRASSIRHIZOMA; ENZYME ASSAY; ENZYME INHIBITION; IC 50; IN VITRO STUDY; POLYACRYLAMIDE GEL ELECTROPHORESIS; STRUCTURE ACTIVITY RELATION;

ACYLATION; DRYOPTERIS; ENZYME INHIBITORS; FATTY ACID SYNTHETASE COMPLEX; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; PHLOROGLUCINOL;

DRYOPTERIDACEAE; DRYOPTERIS CRASSIRHIZOMA;

EID: 33747016347     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.07.018     Document Type: Article

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