5-Alkylated thiazolidinones as follicle-stimulating hormone (FSH) receptor agonists

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 16, 2006, Pages 5729-5741

  Wrobel, Jay ^a   Jetter, James ^a   Kao, Wenling ^a   Rogers, John ^a   Di, Li ^a   Chi, Jamin ^a   Peréz, M Claudia ^a   Chen, Gi Chung ^a   Shen, Emily S ^a  

^a PFIZER INC   (United States)

Author keywords

Follicle stimulating hormone; FSH; FSH receptor agonist; Thiazolidinone

Indexed keywords

CYCLIC AMP RESPONSIVE ELEMENT BINDING PROTEIN; FOLLITROPIN RECEPTOR STIMULATING AGENT; HORMONE RECEPTOR STIMULATING AGENT; LUCIFERASE; THIAZOLIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ALKYLATION; ANIMAL CELL; ARTICLE; CHO CELL; CONTROLLED STUDY; DNA RESPONSIVE ELEMENT; DRUG HYDROLYSIS; DRUG POTENCY; DRUG TOLERABILITY; ENZYME REGULATION; GENE EXPRESSION; GENE OVEREXPRESSION; HORMONAL REGULATION; HORMONE ACTION; IC 50; NONHUMAN; PROTEIN INDUCTION; REPORTER GENE;

ALKYLATION; ANIMALS; CELL LINE; CHO CELLS; CRICETINAE; CYCLIC AMP; FEMALE; FOLLICLE STIMULATING HORMONE; HUMANS; LUCIFERASES; OVARY; RECEPTORS, FSH; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINEDIONES;

CRICETULUS GRISEUS;

EID: 33745608074     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2006.04.012     Document Type: Article

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