Identification and characterization of a selective, nonpeptide follicle-stimulating hormone receptor antagonist

Endocrinology

Volumn 143, Issue 10, 2002, Pages 3822-3829

  Arey, Brian J ^a   Deecher, Darlene C ^a   Shen, Emily S ^b   Stevis, Panayiotis E ^a   Meade Jr , Edwin H ^c   Wrobel, J A Y ^a   Frail, Donald E ^b   López, Francisco J ^c  

^a PFIZER INC   (United States)

^b BRISTOL MYERS SQUIBB   (United States)

^c LIGAND PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

7 [4 [BIS (2 CARBAMOYLETHYL)AMINO] 6 CHLORO 1,3,5 TRIAZIN 2 YLAMINO 4 HYDROXY 3 (4 METHOXYPHENYLAZO)NAPHTHALENE] 2 SULFONIC ACID; FOLLITROPIN; FOLLITROPIN RECEPTOR BINDING INHIBITOR; G PROTEIN COUPLED RECEPTOR; IODINE 125; LUTEINIZING HORMONE; THYROTROPIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BACULOVIRUS; CHO CELL; CONTROLLED STUDY; DRUG ACTIVITY; DRUG IDENTIFICATION; FEMALE; HORMONE INHIBITION; HORMONE RECEPTOR INTERACTION; LIGAND BINDING; NONHUMAN; OVULATION INHIBITION; PRIORITY JOURNAL; RAT; STEROIDOGENESIS;

ANIMALS; BINDING, COMPETITIVE; CELLS, CULTURED; CRICETINAE; EXTRACELLULAR SPACE; FEMALE; FOLLICLE STIMULATING HORMONE; HUMANS; MALE; OVULATION; PROTEIN STRUCTURE, TERTIARY; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, FSH; SULFONIC ACIDS; TRIAZINES;

EID: 0036772776     PISSN: 00137227     EISSN: None     Source Type: Journal    
DOI: 10.1210/en.2002-220372     Document Type: Article

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