Small molecule biaryl FSH receptor agonists. Part 2: Lead optimization via parallel synthesis

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 7, 2004, Pages 1717-1720

  Guo, Tao ^a   Adang, Anton E P ^b   Dong, Guizhen ^a   Fitzpatrick, Dan ^a   Geng, Peng ^a   Ho, Koc Kan ^a   Jibilian, Charles H ^a   Kultgen, Steven G ^a   Liu, Ruiyan ^a   McDonald, Edward ^a   Saionz, Kurt W ^a   Valenzano, Kenneth J ^a   Van Straten, Nicole C R ^b   Xie, Dan ^a   Webb, Maria L ^a  

^a PHARMACOPEIA INC   (United States)

^b NV ORGANON   (Netherlands)

Author keywords

FSH Receptor agonists; Parallel synthesis

Indexed keywords

FOLLICLE STIMULATING HORMONE RECEPTOR AGONIST; HORMONE RECEPTOR STIMULATING AGENT; PIPERAZINEDIONE; UNCLASSIFIED DRUG;

ARTICLE; CYCLIZATION; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; REACTION OPTIMIZATION;

ANIMALS; CHO CELLS; CRICETINAE; PIPERAZINES; RECEPTORS, FSH;

EID: 12144290509     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.01.043     Document Type: Article

References (8)

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