The high throughput screening of neuropeptide FF2 receptor ligands from Korean herbal plant extracts

Peptides

Volumn 27, Issue 5, 2006, Pages 997-1004

  Do, Ernest U ^a   Piao, Long Zhu ^b   Choi, Gyu ^b   Choi, Young Bong ^b   Kang, Tong Mook ^b   Shin, Jaekyoon ^b   Chang, Yung Jin ^a   Nam, Hee Young ^a   Kim, Ho Jin ^a   Kim, Su il ^a  

^a Seoul National University   (South Korea)

^b Sungkyunkwan University   (South Korea)

Author keywords

CRE luciferase reporter assay; Fluorescence polarization; High throughput screening; Neuropeptide FF; Neuropeptide FF2 receptor; Rank order of potency

Indexed keywords

6 BENZOYLOXY 6,7,8,9 TETRAHYDRO 1,2,3,12,13,14 HEXAMETHOXY 7,8 DIMETHYL 7 DIBENZO[A,C]CYCLOOCTENOL; ANTIOBESITY AGENT; ASPARTYLMETHIONINE NEUROPEPTIDE FF; CRE RECOMBINASE; FORSKOLIN; GOMISIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); NALPHA (DIPHENYLACETYL) N (4 HYDROXYBENZYL) DEXTRO ARGININAMIDE; NEUROPEPTIDE FF; NEUROPEPTIDE FF2 RECEPTOR; NEUROPEPTIDE FF2 RECEPTOR AGONIST; NEUROPEPTIDE RECEPTOR; PC 314; PC 315; PEPTIDE; PLANT EXTRACT; PROLYLGLUTAMINYLARGINYLPHENYLALANINAMIDE; SCHIZANDRA CHINENSIS EXTRACT; UNCLASSIFIED DRUG;

ACCURACY; ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING ASSAY; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG ISOLATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SCREENING; ENZYME ASSAY; ETHNOPHARMACOLOGY; FEMALE; FLUORESCENCE POLARIZATION; GENE VECTOR; GENETIC TRANSFECTION; HIGH THROUGHPUT SCREENING; HUMAN; HUMAN TISSUE; IN VITRO STUDY; MEDICINAL PLANT; MICROTITER PLATE ASSAY; NONHUMAN; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN EXPRESSION; RECEPTOR BINDING; REPORTER GENE; REPRODUCIBILITY; SCHISANDRACEAE; SCHIZANDRA CHINENSIS;

COMBINATORIAL CHEMISTRY TECHNIQUES; CYCLOOCTANES; DIOXOLES; DRUG EVALUATION, PRECLINICAL; FLUORESCENCE POLARIZATION; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; KOREA; LIGNANS; MEDICINE, ORIENTAL TRADITIONAL; PEPTIDE LIBRARY; PLANT EXTRACTS; RECEPTORS, NEUROPEPTIDE; SCHISANDRA;

ANIMALIA; SCHISANDRA CHINENSIS; SCHISANDRACEAE;

EID: 33646136254     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.peptides.2005.07.027     Document Type: Article

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