Functional characterization of a human receptor for neuropeptide FF and related peptides

British Journal of Pharmacology

Volumn 133, Issue 1, 2001, Pages 138-144

  Kotani, Masato ^a   Mollereau, Catherine ^b   Detheux, Michel ^c   Le Poul, Emmanuel ^c   Brézillon, Stéphane ^c   Vakili, Jalal ^b   Mazarguil, Honoré ^b   Vassart, Gilbert ^a   Zajac, Jean Marie ^b   Parmentier, Marc ^a  

^a UNIVERSITÉ LIBRE DE BRUXELLES   (Belgium)

^b INSTITUT DE PHARMACOLOGIE ET DE BIOLOGIE STRUCTURALE   (France)

^c Euroscreen SA   (Belgium)

Author keywords

Aequorin assay; G protein coupled receptor; Neuropeptide AF; Neuropeptide FF; Orphan receptor

Indexed keywords

CYCLIC AMP; FORSKOLIN; G PROTEIN COUPLED RECEPTOR; MESSENGER RNA; NEUROPEPTIDE FF; PEPTIDE DERIVATIVE; PERTUSSIS TOXIN;

ANIMAL CELL; ARTICLE; CHO CELL; CONTROLLED STUDY; DOSE RESPONSE; DRUG POTENCY; DRUG RECEPTOR BINDING; FEMALE; GENE EXPRESSION; NEUROMODULATION; NONHUMAN; NUCLEOTIDE SEQUENCE; PAIN THRESHOLD; PRIORITY JOURNAL; RECEPTOR AFFINITY; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION;

EID: 0034982423     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704038     Document Type: Article

References (30)

1. Characterization and localization of a putative morphine-modulating peptide, FLFQPQRFamide, in the rat spinal cord: Biochemical and immunocytochemical studies
2. Multiple charged and aromatic residues in CCR5 amino-terminal domain are involved in high affinity binding of both chemokines and HIV-1 env protein
3. Identification and characterization of two G protein-coupled receptors for neuropeptide FF
4. Sequence and tissue distribution of a novel G protein-coupled receptor expressed prominently in human placenta
5. Natural proteolytic processing of hemofiltrate CC chemokine 1 generates a potent CC chemokine receptor (CCR)1 and CCR5 agonist with anti-HIV properties
6. Characterization of a potent agonist for NPFF receptors: Binding study in rat spinal cord membranes
7. Effects of neuropeptide FF analogs on morphine analgesia in the nucleus raphe dorsalis
8. 3]NPFF
9. Receptor for the pain modulatory neuropeptide FF and AF is an orphan G protein-coupled receptor
10. Antisense oligonucleotides to human SQA-neuropeptide FF decrease morphine tolerance and dependence in mice
11. Neuropeptide FF receptors of mouse olfactory bulb: Binding properties and stimulation of adenylate cyclase activity
12. 125I]EYF: A new high affinity radioligand to Neuropeptide FF receptors
13. Antinociceptive effects of intrathecally administered F8Famide and FMRFamide in the rat
14. 3]NPFF
15. New neuropeptides containing carboxy-terminal RFamide and their receptor in mammals
16. Immunohistochemical distribution and partial characterization of FLFQPQRFamide-like peptides in the central nervous system of rats
17. Modulation of human lymphocyte proliferation by FLFQPQRFamide, a FMRFamide-like peptide with anti-opiate properties
18. Distribution and characterization of neuropeptide FF-like immunoreactivity in the rat nervous system with a monoclonal antibody
19. 2-like peptide
20. Biphasic effect on nociceptin and antiopiate activity of neuropeptide FF (FLFQPQRFamide) in the rat
21. Neuropeptide FF, a mammalian neuropeptide with multiple functions
22. Neuropeptide FF receptors: Structure-activity relationship and effect of morphine
23. Modulating of neuropeptide FF receptors by guanine nucleotides and cations in membranes of rat brain and spinal cord
24. A human gene encoding morphine modulating peptides related to NPFF and FMRFamide
25. Are neuropeptides FF and SF neurotransmitters in the rat?
26. Neuropeptide FF, pain and analgesia
27. A simple direct assay for cyclic AMP in plasma and other biological samples using an improved competitive protein binding technique
28. Gene for pain modulatory neuropeptide NPFF: Induction in spinal cord by noxious stimuli
29. Isolation, sequencing, synthesis, and pharmacological characterization of the two brain neuropeptides that modulate the action of morphine
30. Neuropeptide FF receptors