Neamine derivatives having a nucleobase with a lysine or an arginine as a linker, their synthesis and evaluation as potential inhibitors for HIV TAR-Tat

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 8, 2006, Pages 2799-2809

  Yajima, Saki ^a   Shionoya, Hirohito ^a   Akagi, Takashi ^a   Hamasaki, Keita ^a  

^a SHIBAURA INSTITUTE OF TECHNOLOGY   (Japan)

Author keywords

Aminoglycoside; Drug design; HIV TAR; HIV Tat; Inhibition; Neamine

Indexed keywords

ARGININE DERIVATIVE; LYSINE DERIVATIVE; NEAMINE; NUCLEIC ACID BASE; TRANSACTIVATOR PROTEIN;

ARTICLE; DRUG SCREENING; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS; PROTEIN INTERACTION; STEREOCHEMISTRY;

AMINO ACID SEQUENCE; AMINOGLYCOSIDES; ANTI-HIV AGENTS; ARGININE; FRAMYCETIN; GENE PRODUCTS, TAT; LYSINE; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR SEQUENCE DATA; SPECTROMETRY, FLUORESCENCE;

HUMAN IMMUNODEFICIENCY VIRUS;

EID: 33644769091     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.11.056     Document Type: Article

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