-
4
-
-
0001050065
-
-
(b) Chavez-Noriega, L. E.; Schaffhauser, H.; Campbell, U. C. Current Drug Targets: CNS & Neurological Disorder 2002, 7, 261.
-
(2002)
Current Drug Targets: CNS & Neurological Disorder
, vol.7
, pp. 261
-
-
Chavez-Noriega, L.E.1
Schaffhauser, H.2
Campbell, U.C.3
-
5
-
-
0032834028
-
-
(c) Schoepp, D. D.; Jane, D. E.; Monn, J. A. Neuropharmacology 1999, 38, 1431.
-
(1999)
Neuropharmacology
, vol.38
, pp. 1431
-
-
Schoepp, D.D.1
Jane, D.E.2
Monn, J.A.3
-
6
-
-
0035282715
-
-
(d) De Blasi, A.; Conn, P. J.; Pin, J.-P.; Nicoletti, F. TRENDS in Pharmacological Sciences 2001, 22, 114. For structure basis of mGluR recognition;
-
(2001)
TRENDS in Pharmacological Sciences
, vol.22
, pp. 114
-
-
De Blasi, A.1
Conn, P.J.2
Pin, J.-P.3
Nicoletti, F.4
-
7
-
-
0034718925
-
-
(e) Kunishima, N.; Shimada, Y.; Tsuji, Y.; Sato, T.; Yamamoto, M.; Kumasaka, T.; Nakanishi, S.; Jingami, H.; Morikawa, K. Nature 2000, 407, 971.
-
(2000)
Nature
, vol.407
, pp. 971
-
-
Kunishima, N.1
Shimada, Y.2
Tsuji, Y.3
Sato, T.4
Yamamoto, M.5
Kumasaka, T.6
Nakanishi, S.7
Jingami, H.8
Morikawa, K.9
-
8
-
-
0037130210
-
-
Bertrand, H.-O.; Bessis, A.-S.; Pin, J.-P.; Acher, F. C. J. Med. Chem. 2002, 45, 3171.
-
(2002)
J. Med. Chem.
, vol.45
, pp. 3171
-
-
Bertrand, H.-O.1
Bessis, A.-S.2
Pin, J.-P.3
Acher, F.C.4
-
9
-
-
15644369847
-
-
(a) Monn, J. A.; Valli, M. J.; Massey, S. M.; Wright, R. A.; Salhoff, C. R.; Johnson, B. G.; Howe, T.; Alt, C. A.; Rhodes, G. A.; Robey, R. L.; Griffey, K. R.; Tizzano, J. P.; Kallman, M. J.; Helton, D. R.; Schoepp, D. D. J. Med. Chem. 1997, 40, 528.
-
(1997)
J. Med. Chem.
, vol.40
, pp. 528
-
-
Monn, J.A.1
Valli, M.J.2
Massey, S.M.3
Wright, R.A.4
Salhoff, C.R.5
Johnson, B.G.6
Howe, T.7
Alt, C.A.8
Rhodes, G.A.9
Robey, R.L.10
Griffey, K.R.11
Tizzano, J.P.12
Kallman, M.J.13
Helton, D.R.14
Schoepp, D.D.15
-
10
-
-
0033602516
-
-
(b) Monn, J. A.; Valli, M. J.; Massey, S. M.; Hansen, M. M.; Kress, T. J.; Wepsiec, J. P.; Harkness, A. R.; Grutsch, J. L.; Wright, R. A.; Johnson, B. G.; Andis, S. L.; Kingston, A.; Tomlison, R.; Lewis, R.; Griffey, K. R.; Tizzano, J. P.; Schoepp, D. D. J. Med. Chem. ibid. 1999, 42, 1027.
-
(1999)
J. Med. Chem.
, vol.42
, pp. 1027
-
-
Monn, J.A.1
Valli, M.J.2
Massey, S.M.3
Hansen, M.M.4
Kress, T.J.5
Wepsiec, J.P.6
Harkness, A.R.7
Grutsch, J.L.8
Wright, R.A.9
Johnson, B.G.10
Andis, S.L.11
Kingston, A.12
Tomlison, R.13
Lewis, R.14
Griffey, K.R.15
Tizzano, J.P.16
Schoepp, D.D.17
-
11
-
-
0037101811
-
-
Collado, I.; Pedregal, C.; Mazón, A.; Espinosa, J. F.; Blanco-Urgoiti, J.; Schoepp, D. D.; Wright, R. A.; Johnson, B. G.; Kingston, A. E. J. Med. Chem. 2002, 45, 3619.
-
(2002)
J. Med. Chem.
, vol.45
, pp. 3619
-
-
Collado, I.1
Pedregal, C.2
Mazón, A.3
Espinosa, J.F.4
Blanco-Urgoiti, J.5
Schoepp, D.D.6
Wright, R.A.7
Johnson, B.G.8
Kingston, A.E.9
-
14
-
-
0034649605
-
-
Nakazato, A.; Kumagai, T.; Sakagami, K.; Yoshikawa, R.; Suzuki, Y.; Chaki, S.; Ito, H.; Nakanishi, S.; Okuyama, S., J. Med. Chem. 2000, 43, 4893.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 4893
-
-
Nakazato, A.1
Kumagai, T.2
Sakagami, K.3
Yoshikawa, R.4
Suzuki, Y.5
Chaki, S.6
Ito, H.7
Nakanishi, S.8
Okuyama, S.9
-
16
-
-
0031579430
-
-
(b) Dominguez, C.; Ezquerra, J.; Prieto, L.; Espada, M.; Pedregal, C. Tetrahedron: Asymmetry 1997, 8, 511. See also 5a.
-
(1997)
Tetrahedron: Asymmetry
, vol.8
, pp. 511
-
-
Dominguez, C.1
Ezquerra, J.2
Prieto, L.3
Espada, M.4
Pedregal, C.5
-
17
-
-
0037863192
-
-
Ohfune, Y.; Demura, T.; Iwama, S.; Matsuda, H.; Namba, K.; Shimamoto, K.; Shinada, T. Tetrahedron Lett. 2003, 44, 5431.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 5431
-
-
Ohfune, Y.1
Demura, T.2
Iwama, S.3
Matsuda, H.4
Namba, K.5
Shimamoto, K.6
Shinada, T.7
-
18
-
-
1642443189
-
-
Wong, A.; Welsh, C. J.; Kuethe, J. T.; Vazquez, E.; Shaimi, M.; Henderson, D.; Davies, I. W.; Hughes, D. L. Org. Biomol. Chem. 2004, 2, 168.
-
(2004)
Org. Biomol. Chem.
, vol.2
, pp. 168
-
-
Wong, A.1
Welsh, C.J.2
Kuethe, J.T.3
Vazquez, E.4
Shaimi, M.5
Henderson, D.6
Davies, I.W.7
Hughes, D.L.8
-
19
-
-
12344335218
-
-
New synthetic method for diazo ketones without using diazomethane equivalents has been reported: Bio, M. M.; Javadi, G.; Song, Z. J. Synthesis 2005, 19.
-
(2005)
Synthesis
, pp. 19
-
-
Bio, M.M.1
Javadi, G.2
Song, Z.J.3
-
20
-
-
85039348405
-
-
Int. Appl. PCT, WO 2002000595
-
Nakazako, A.; Kumagai, T.; Sakagami, K.; Taguchi, T. Int. Appl. PCT, WO 2002000595, 2002.
-
(2002)
-
-
Nakazako, A.1
Kumagai, T.2
Sakagami, K.3
Taguchi, T.4
-
21
-
-
7044260863
-
-
Zhang, F.; Song, Z. J.; Tschaen, D.; Volante, R. P. Org. Lett. 2004, 6, 3775.
-
(2004)
Org. Lett.
, vol.6
, pp. 3775
-
-
Zhang, F.1
Song, Z.J.2
Tschaen, D.3
Volante, R.P.4
-
23
-
-
33746494993
-
-
Ito, Y.; Hirao, T.; Saegusa, T. J. Org. Chem. 1978, 43, 1011.
-
(1978)
J. Org. Chem.
, vol.43
, pp. 1011
-
-
Ito, Y.1
Hirao, T.2
Saegusa, T.3
-
24
-
-
85039344530
-
-
Unpublished results
-
Unpublished results.
-
-
-
-
25
-
-
0028854518
-
-
Interesting stereochemistry has been reported; Otera, J.; Fujita, Y.; Fukuzumi, S.; Hirai, K.-I.; Gu, J.-H.; Nakai, T. Tetrahedron Lett. 1995, 36, 95.
-
(1995)
Tetrahedron Lett.
, vol.36
, pp. 95
-
-
Otera, J.1
Fujita, Y.2
Fukuzumi, S.3
Hirai, K.-I.4
Gu, J.-H.5
Nakai, T.6
-
26
-
-
25444486184
-
-
Tan, L.; Yasuda, N.; Yoshikawa, N.; Hartner, F. W.; Eng, K. K.; Leonard, W. R.; Tsay, F.-R.; Volante, R. P.; Tillyer, R. D. J. Org. Chem. 2005, 70, 8027.
-
(2005)
J. Org. Chem.
, vol.70
, pp. 8027
-
-
Tan, L.1
Yasuda, N.2
Yoshikawa, N.3
Hartner, F.W.4
Eng, K.K.5
Leonard, W.R.6
Tsay, F.-R.7
Volante, R.P.8
Tillyer, R.D.9
-
27
-
-
0035959461
-
-
Saito, A.; Ito, H.; Taguchi, T. Tetrahedron 2001, 57, 7487.
-
(2001)
Tetrahedron
, vol.57
, pp. 7487
-
-
Saito, A.1
Ito, H.2
Taguchi, T.3
-
29
-
-
4444373880
-
-
Yoshikawa, N.; Tan, L.; Yasuda, N.; Volante, R.P.; Tillyer, R. D. Tetrahedron Lett. 2004, 45, 7261.
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 7261
-
-
Yoshikawa, N.1
Tan, L.2
Yasuda, N.3
Volante, R.P.4
Tillyer, R.D.5
-
30
-
-
0001215705
-
-
For Lewis acid assisted epoxide opening with enolates; see: (a) Taylor, S. K.; Fried, J. A.; Grassl, Y. N.; Marolewski, A. E.; Pelton, E. A.; Poel, T.-J.; Rezanka, D. S.; Whittaker, M. R. J. Org. Chem. 1993, 58, 7304.
-
(1993)
J. Org. Chem.
, vol.58
, pp. 7304
-
-
Taylor, S.K.1
Fried, J.A.2
Grassl, Y.N.3
Marolewski, A.E.4
Pelton, E.A.5
Poel, T.-J.6
Rezanka, D.S.7
Whittaker, M.R.8
-
31
-
-
0001435803
-
-
(b) Crotti, P.; Bussolo, V. D.; Favero, L.; Pineschi, M.; Pasero, M. J. Org. Chem. ibid. 1996, 61, 9548.
-
(1996)
J. Org. Chem.
, vol.61
, pp. 9548
-
-
Crotti, P.1
Bussolo, V.D.2
Favero, L.3
Pineschi, M.4
Pasero, M.5
-
32
-
-
0033617237
-
-
(c) Crotti, P.; Bussolo, V. D.; Favero, L.; Macchia, F.; Pineschi, M.; Napolitano, E. Tetrahedron 1999, 55, 5853.
-
(1999)
Tetrahedron
, vol.55
, pp. 5853
-
-
Crotti, P.1
Bussolo, V.D.2
Favero, L.3
Macchia, F.4
Pineschi, M.5
Napolitano, E.6
-
33
-
-
0037022458
-
-
(d) Hojo, M.; Sakata, K.; Maimaiti, X.; Ueno, J.; Nishikori, H.; Hosomi, A. Chem. Lett. 2002, 142.
-
(2002)
Chem. Lett.
, pp. 142
-
-
Hojo, M.1
Sakata, K.2
Maimaiti, X.3
Ueno, J.4
Nishikori, H.5
Hosomi, A.6
-
34
-
-
0015928584
-
-
Partridge, J. J.; Chadha, N. K.; Uskokovic, M. R. J. Am. Chem. Soc. 1973, 95, 7171;
-
(1973)
J. Am. Chem. Soc.
, vol.95
, pp. 7171
-
-
Partridge, J.J.1
Chadha, N.K.2
Uskokovic, M.R.3
-
35
-
-
31344480905
-
-
Organic Syntheses 1985, 63, 44.
-
(1985)
Organic Syntheses
, vol.63
, pp. 44
-
-
-
36
-
-
0000458209
-
-
For directed epoxidation, see: Hoveyda, A. H.; Evans, D. A.; Fu, G. C. Chem. Rev. 1993, 93, 1307.
-
(1993)
Chem. Rev.
, vol.93
, pp. 1307
-
-
Hoveyda, A.H.1
Evans, D.A.2
Fu, G.C.3
-
37
-
-
0034699797
-
-
In acyclic cases, facile cyclopropanation reaction without Lewis acids was reported; Agami, C.; Couty, F.; Evano, G. Tetrahedron Lett. 2000, 41, 8301.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 8301
-
-
Agami, C.1
Couty, F.2
Evano, G.3
-
38
-
-
0029980473
-
-
Cai, D.; Hughes, D. L.; Verhoeven, T. R. Tetrahedron Lett. 1996, 37, 2537.
-
(1996)
Tetrahedron Lett.
, vol.37
, pp. 2537
-
-
Cai, D.1
Hughes, D.L.2
Verhoeven, T.R.3
-
39
-
-
85039357526
-
-
Unpublished results
-
Unpublished results.
-
-
-
-
40
-
-
0000169587
-
-
Tsunoda, T.; Suzuki, M.; Noyori, R. Tetrahedron Lett. 1980, 21, 1357.
-
(1980)
Tetrahedron Lett.
, vol.21
, pp. 1357
-
-
Tsunoda, T.1
Suzuki, M.2
Noyori, R.3
-
41
-
-
0034641473
-
-
Postel, D.; Nguyen Van Nhien, A.; Pillon, M.; Villa, P.; Ronco, G. Tetrahedron Lett. 2000, 41, 6403.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 6403
-
-
Postel, D.1
Nguyen Van Nhien, A.2
Pillon, M.3
Villa, P.4
Ronco, G.5
|