DNA sequence recognition in the minor groove by hairpin pyrrole polyamide-Hoechst 33258 analogue conjugate

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 14, 2004, Pages 3803-3807

  Reddy, Putta Mallikarjuna ^a   Dexter, Rachel ^a   Bruice, Thomas C ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [5 (4 METHYL 1 PIPERAZINYL)[2,5' BI 1H BENZIMIDAZOL] 2' YL]PHENOL; DOUBLE STRANDED DNA; POLYAMIDE; PYRROLE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CHEMICAL REACTION KINETICS; DNA SEQUENCE; DRUG CONJUGATION; DRUG SYNTHESIS; MELTING POINT; MOLECULAR RECOGNITION; SOLID PHASE EXTRACTION; SPECTROFLUOROMETRY; TITRIMETRY;

BASE SEQUENCE; BINDING SITES; BISBENZIMIDE; DNA; MOLECULAR STRUCTURE; NUCLEIC ACID CONFORMATION; NYLONS; PYRROLES; SPECTROMETRY, FLUORESCENCE; TEMPERATURE; TITRIMETRY;

EID: 2942538217     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.04.089     Document Type: Article

References (28)

1. Latchman D.S. Gene regulation: a eukaryotic perspective. 3rd ed. 1998;Stanley Thornes, Cheltenham
2. Bailly C., Chaires J.B. Bioconjugate Chem. 9:1998;513
3. Reddy B.S.P., Sondhi S.M., Lown J.W. Pharmacol. Ther. 84:1999;1
4. Dervan P.B. Bioorg. Med. Chem. 9:2001;2215
5. Neidle S. Nat. Prod. Rep. 18:2001;291
6. Chiang S.-Y., Bruice T.C., Azizkhan J.C., Gawron L., Beerman T.A. Proc. Natl. Acad. Sci. U.S.A. 94:1997;2811
7. He G.X., Browne K.A., Blasko A., Bruice T.C. J. Am. Chem. Soc. 116:1994;3716
8. Browne K.A., He G.X., Bruice T.C. J. Am. Chem. Soc. 115:1993;7072
9. Dervan P.B., Edelson B.S. Curr. Opin. Struct. Biol. 13:2003;284
10. Dervan P.B., Burli R.W. Curr. Opin. Chem. Biol. 3:1999;688
11. Gottesfeld J.M., Neeley L., Trauger J.W., Baird E.E., Dervan P.B. Nature. 387:1997;202
12. Mapp A.M., Ansari A.Z., Ptashne M., Dervan P.B. Proc. Natl. Acad. Sci. U.S.A. 97:2000;3930
13. Chiang S.Y., Burli R.W., Benz C.C., Gawron L., Scott G.K., Dervan P.B., Beerman T.A. J. Biol. Chem. 275:2000;24246
14. Holmquist G. Chromosoma. 49:1975;333
15. Arndt-Jovin D.J., Jovin T.M. Cytometry. 11:1990;80
16. Frau S., Bernadou J., Meunier B. Bull. Soc. Chim. Fr. 133:1996;1053
17. Satz A.L., Bruice T.C. J. Am. Chem. Soc. 123:2001;2469
18. Satz A.L., Bruice T.C. Bioorg. Med. Chem. 10:2002;241
19. Reddy P.M., Jindra P.T., Satz A.L., Bruice T.C. J. Am. Chem. Soc. 125:2003;7843
20. White C.M., Satz A.L., Bruice T.C., Beerman T.A. Proc. Natl. Acad. Sci. U.S.A. 98:2001;10590
21. White C.M., Satz A.L., Gawron L.S., Bruice T.C., Beerman T.A. Biochim. Biophys. Acta. 1574:2001;100
22. Wurtz N.R., Turner J.M., Baird E.E., Dervan P.B. Org. Lett. 3:2001;1201
23. Reddy P.M., Bruice T.C. J. Am. Chem. Soc. 126:2004;3736
24. Loontiens F.G., Regenfuss P., Zechel A., Dumortier L., Clegg R.M. Biochemistry. 29:1990;9029
25. Bostock-Smith C.E., Searle M.S. Nucl. Acids Res. 27:1999;1619
26. Haq I., Ladbury J.E., Chowdhry B.Z., Jenkins T.C., Chaires J.B. J. Mol. Biol. 271:1997;244
27. Loontiens F.G., McLaughlin L.W., Diekmann S., Clegg R.M. Biochemistry. 30:1991;182
28. Satz A.L., Bruice T.C. Bioorg. Med. Chem. 8:2000;1871