Synthesis and evaluation of a potent and selective cell-permeable p300 histone acetyltransferase inhibitor

Journal of the American Chemical Society

Volumn 127, Issue 49, 2005, Pages 17182-17183

  Zheng, Yujun ^a   Balasubramanyam, Karanam ^a   Cebrat, Marek ^a   Buck, Donald ^a   Guidez, Fabien ^b   Zelent, Arthur ^b   Alani, Rhoda M ^a   Cole, Philip A ^a  

^a JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b INSTITUTE OF CANCER RESEARCH   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; HISTONE ACETYLTRANSFERASE INHIBITOR; PROTEIN P300; UNCLASSIFIED DRUG;

ACETYLATION; ARTICLE; CONTROLLED STUDY; DISULFIDE BOND; DRUG POTENCY; DRUG SPECIFICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; TRANSCRIPTION REGULATION;

EID: 29044440879     PISSN: 00027863     EISSN: None     Source Type: Journal    
DOI: 10.1021/ja0558544     Document Type: Article

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