Inhibitory modulation of ATP-sensitive potassium channels by gallate-ester moiety of (-)-epigallocatechin-3-gallate

Biochemical Pharmacology

Volumn 70, Issue 11, 2005, Pages 1560-1567

  Baek, Won Ki ^a   Jang, Byeong Churl ^a   Jun, Hee Lim ^a   Kwon, Taeg Kyu ^a   Lee, Hyun Young ^a   Cho, Chi Heum ^a   Kim, Dae Kwang ^a   Shin, Dong Hoon ^a   Park, Jong Gu ^a   Lim, Jeong Geun ^a   Bae, Ji Hyun ^a   Bae, Jae Hoon ^a   Sun, Kyun Yoo ^b   Park, Won Kyun ^a   Song, Dae Kyu ^a  

^a Keimyung University   (South Korea)

^b Joongbu University   (South Korea)

Author keywords

ATP sensitive potassium channel; EGCG; Gallate ester moiety; Kir6.2; Pancreatic cell; Xenopus oocyte

Indexed keywords

ADENOSINE TRIPHOSPHATE; EPICATECHIN; EPICATECHIN 3 GALLATE; EPIGALLOCATECHIN; EPIGALLOCATECHIN GALLATE; GALLIC ACID DERIVATIVE; GREEN TEA EXTRACT; INWARDLY RECTIFYING POTASSIUM CHANNEL SUBUNIT KIR6.2; POLYPHENOL DERIVATIVE; POTASSIUM CHANNEL; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; DRUG MECHANISM; DRUG POTENCY; DRUG STRUCTURE; FEMALE; IC 50; MOLECULAR BIOLOGY; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PRIORITY JOURNAL; XENOPUS;

ADENOSINE TRIPHOSPHATE; ANIMALS; CATECHIN; CELL MEMBRANE; ION CHANNEL GATING; ISLETS OF LANGERHANS; MEMBRANE POTENTIALS; MOLECULAR STRUCTURE; OOCYTES; POTASSIUM CHANNEL BLOCKERS; POTASSIUM CHANNELS, INWARDLY RECTIFYING; PROTEIN SUBUNITS; STRUCTURE-ACTIVITY RELATIONSHIP; XENOPUS LAEVIS;

EID: 27544447337     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2005.09.005     Document Type: Article

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