-
1
-
-
2142653053
-
A homogeneous fluorescence polarization assay adaptable for a range of protein scrine/threonine and tyrosine kinases
-
Gaudet EA, Huang K-S, Zhang Y, Huang W, Mark D, Sportsman JR: A homogeneous fluorescence polarization assay adaptable for a range of protein scrine/threonine and tyrosine kinases. J Biomol Screen 2003;8:164-175.
-
(2003)
J. Biomol. Screen.
, vol.8
, pp. 164-175
-
-
Gaudet, E.A.1
Huang, K.-S.2
Zhang, Y.3
Huang, W.4
Mark, D.5
Sportsman, J.R.6
-
2
-
-
2442583662
-
High-throughput screening with immobilized metal ion affinity-based fluorescence polarization detection, a homogenous assay for protein kinases
-
Loomans EE, van Doornmalen AM, Wat JW, Zaman GJ: High-throughput screening with immobilized metal ion affinity-based fluorescence polarization detection, a homogenous assay for protein kinases. Assay Drug Dev Technol 2003;1:445-453.
-
(2003)
Assay Drug Dev. Technol.
, vol.1
, pp. 445-453
-
-
Loomans, E.E.1
van Doornmalen, A.M.2
Wat, J.W.3
Zaman, G.J.4
-
3
-
-
2442585687
-
Development of a fluorescence polarization Akt serine/threonine kinase assay using an immobilized metal ion affinity-based technology
-
Turek-Etienne TC, Kober TP, Stafford JM, Bryant RW: Development of a fluorescence polarization Akt serine/threonine kinase assay using an immobilized metal ion affinity-based technology. Assay Drug Dev Technol 2003; 1:545-553.
-
(2003)
Assay Drug Dev. Technol.
, vol.1
, pp. 545-553
-
-
Turek-Etienne, T.C.1
Kober, T.P.2
Stafford, J.M.3
Bryant, R.W.4
-
4
-
-
0038284889
-
Competitive fluorescence polarization assays for the detection of phosphoinositide kinase and phosphatase activity
-
Drees BE, Weipert A, Hudson H, Ferguson CG, Chakravarty L, Prestwich GD: Competitive fluorescence polarization assays for the detection of phosphoinositide kinase and phosphatase activity. Comb Chem High Throughput Screen 2003;6:321-330.
-
(2003)
Comb. Chem. High Throughput Screen.
, vol.6
, pp. 321-330
-
-
Drees, B.E.1
Weipert, A.2
Hudson, H.3
Ferguson, C.G.4
Chakravarty, L.5
Prestwich, G.D.6
-
5
-
-
18644384952
-
M. An evaluation of fluorescence polarization and lifetime discriminated polarization for high throughput screening of serine/threonine kinases
-
Fowler A, Swift D, Longman E, Acornley A, Hemsley P, Murray D, Unitt J, Dale I, Sullivan E, Coldwell M: An evaluation of fluorescence polarization and lifetime discriminated polarization for high throughput screening of serine/threonine kinases. Anal Biochem 2002;308:223-231.
-
(2002)
Anal. Biochem.
, vol.308
, pp. 223-231
-
-
Fowler, A.1
Swift, D.2
Longman, E.3
Acornley, A.4
Hemsley, P.5
Murray, D.6
Unitt, J.7
Dale, I.8
Sullivan, E.9
Coldwell, M.10
-
6
-
-
0035991330
-
Comparison of assay technologies for a tyrosine kinase assay generates different results in high throughput screening
-
Sills MA, Weiss D, Pham Q, Schweitzer R, Wu X, Wu JJ: Comparison of assay technologies for a tyrosine kinase assay generates different results in high throughput screening. J Biomol Screen 2002;7:191-214.
-
(2002)
J. Biomol. Screen.
, vol.7
, pp. 191-214
-
-
Sills, M.A.1
Weiss, D.2
Pham, Q.3
Schweitzer, R.4
Wu, X.5
Wu, J.J.6
-
7
-
-
0346279807
-
Evaluation of fluorescent compound interference in 4 fluorescence polarization assays: 2 kinases, 1 protease, and 1 phosphatase
-
Turek-Etienne TC, Small EC, Soh SC, Xin TA, Gaitonde PV, Barrabee EB, Hart RF, Bryant RW: Evaluation of fluorescent compound interference in 4 fluorescence polarization assays: 2 kinases, 1 protease, and 1 phosphatase. J Biomol Screen 2003;8:176-184.
-
(2003)
J. Biomol. Screen.
, vol.8
, pp. 176-184
-
-
Turek-Etienne, T.C.1
Small, E.C.2
Soh, S.C.3
Xin, T.A.4
Gaitonde, P.V.5
Barrabee, E.B.6
Hart, R.F.7
Bryant, R.W.8
-
8
-
-
0033003760
-
A simple statistical parameter for use in evaluation and validation of high throughput screening assays
-
Zhang JH, Chung TD, Oldenburg KR: A simple statistical parameter for use in evaluation and validation of high throughput screening assays. J Biomol Screen 1999;4:67-73.
-
(1999)
J. Biomol. Screen.
, vol.4
, pp. 67-73
-
-
Zhang, J.H.1
Chung, T.D.2
Oldenburg, K.R.3
-
9
-
-
0001310375
-
Fluorescence polarization
-
Devlin JP (ed.), Marcel Dekker, New York
-
Sportsman JR, Lee SL, Dilley H, Bukar R: Fluorescence polarization. In: High Throughput Screening: the Discovery of Bioactive Substances. Devlin JP (ed.), pp. 389-399. Marcel Dekker, New York, 1997.
-
(1997)
High Throughput Screening: The Discovery of Bioactive Substances
, pp. 389-399
-
-
Sportsman, J.R.1
Lee, S.L.2
Dilley, H.3
Bukar, R.4
-
10
-
-
0033778265
-
Impact of a red-shifted dye label for high throughput fluorescence polarization assays of G protein-coupled receptors
-
Banks P, Gosselin M, Prystay L: Impact of a red-shifted dye label for high throughput fluorescence polarization assays of G protein-coupled receptors. J Biomol Screen 2000; 5:329-334.
-
(2000)
J. Biomol. Screen.
, vol.5
, pp. 329-334
-
-
Banks, P.1
Gosselin, M.2
Prystay, L.3
-
11
-
-
2442521478
-
Use of red-shifted dyes in a fluorescence polarization AKT kinase assay for detection of biological activity in natural product extracts
-
Turek-Etienne TC, Lei M, Terracciano JS, Langsdorf EF, Bryant RW, Hart RF, Horan AC: Use of red-shifted dyes in a fluorescence polarization AKT kinase assay for detection of biological activity in natural product extracts. J Biomol Screen 2004;9:52-61.
-
(2004)
J. Biomol. Screen.
, vol.9
, pp. 52-61
-
-
Turek-Etienne, T.C.1
Lei, M.2
Terracciano, J.S.3
Langsdorf, E.F.4
Bryant, R.W.5
Hart, R.F.6
Horan, A.C.7
-
12
-
-
1842775922
-
Miniaturization of fluorescence polarization receptor-binding assays using Cy-Dye-labeled ligands
-
Harris A, Cox S, Burns D, Norey C: Miniaturization of fluorescence polarization receptor-binding assays using Cy-Dye-labeled ligands. J Biomol Screen 2003;8:410-420.
-
(2003)
J. Biomol. Screen.
, vol.8
, pp. 410-420
-
-
Harris, A.1
Cox, S.2
Burns, D.3
Norey, C.4
-
13
-
-
0033773937
-
Fluorescence polarization and anisotropy in high throughput screening: Perspectives and primer
-
Owicki JC: Fluorescence polarization and anisotropy in high throughput screening: perspectives and primer. J Biomol Screen 2000;5:297-306.
-
(2000)
J. Biomol. Screen.
, vol.5
, pp. 297-306
-
-
Owicki, J.C.1
-
14
-
-
2442457987
-
Evaluation of compound interference in immobilized metal ion affinity-based fluorescence polarization detection with a four million member compound collection
-
Beasley JR, Dunn DA, Walker TL, Parlato SM, Lehrach JM, Auld DS: Evaluation of compound interference in immobilized metal ion affinity-based fluorescence polarization detection with a four million member compound collection. Assay Drug Dev Technol 2003;1:455-459.
-
(2003)
Assay Drug Dev. Technol.
, vol.1
, pp. 455-459
-
-
Beasley, J.R.1
Dunn, D.A.2
Walker, T.L.3
Parlato, S.M.4
Lehrach, J.M.5
Auld, D.S.6
-
15
-
-
0023022190
-
Selective adsorption of phosphoproteins on gel-immobilized ferric chelate
-
Musuzynska G, Andersson L, Porath J: Selective adsorption of phosphoproteins on gel-immobilized ferric chelate. Biochemistry 1986;25:6850-6853.
-
(1986)
Biochemistry
, vol.25
, pp. 6850-6853
-
-
Musuzynska, G.1
Andersson, L.2
Porath, J.3
-
16
-
-
2442501720
-
Determining appropriate substrate conversion for enzymatic assays in high-throughput screening
-
Wu G, Yuan Y, Hodge CN: Determining appropriate substrate conversion for enzymatic assays in high-throughput screening. J Biomol Screen 2003;8:694-700.
-
(2003)
J. Biomol. Screen.
, vol.8
, pp. 694-700
-
-
Wu, G.1
Yuan, Y.2
Hodge, C.N.3
-
17
-
-
2442478704
-
Assay tutorial: Nonradioactive FP-based IMAP assay for kinases, phosphatases, and phosphodiesterases
-
Adams C, Gaudet EA, Boge A: Assay tutorial: Nonradioactive FP-based IMAP assay for kinases, phosphatases, and phosphodiesterases. Genet Eng News 2003;23:38-39.
-
(2003)
Genet. Eng. News
, vol.23
, pp. 38-39
-
-
Adams, C.1
Gaudet, E.A.2
Boge, A.3
-
18
-
-
2442449561
-
Development of a fluorescence polarization bead-based coupled assay to target different activity/conformation states of a protein kinase
-
(in press)
-
Lu Z, Yin Z, James L, Syto R, Stafford JM, Koseoglu S, Mayhood T, Myers J, Windsor W, Kirschmeier P, Samatar A, Malcolm B, Turek-Etienne TC, Kumar CC: Development of a fluorescence polarization bead-based coupled assay to target different activity/conformation states of a protein kinase. J Biomol Screen 2004 (in press).
-
(2004)
J. Biomol. Screen.
-
-
Lu, Z.1
Yin, Z.2
James, L.3
Syto, R.4
Stafford, J.M.5
Koseoglu, S.6
Mayhood, T.7
Myers, J.8
Windsor, W.9
Kirschmeier, P.10
Samatar, A.11
Malcolm, B.12
Turek-Etienne, T.C.13
Kumar, C.C.14
-
19
-
-
0141788346
-
STI-571: An anticancer protein-tyrosine kinase inhibitor
-
Roskoski R Jr: STI-571: an anticancer protein-tyrosine kinase inhibitor. Biochem Biophys Res Commun 2003;309: 709-717.
-
(2003)
Biochem. Biophys. Res. Commun.
, vol.309
, pp. 709-717
-
-
Roskoski Jr., R.1
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