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Volumn 7, Issue 17, 2005, Pages 3749-3752

Directed ortho lithiation of N-alkylphenylaziridines

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EID: 24044445511     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol051412l     Document Type: Article
Times cited : (67)

References (53)
  • 1
    • 0002307974 scopus 로고
    • For extensive reviews on ortho lithiation and for various DMGs, see: (a) Gschwend, H. W.; Rodriguez, H. R. Org. React. 1979, 26, 1-360.
    • (1979) Org. React. , vol.26 , pp. 1-360
    • Gschwend, H.W.1    Rodriguez, H.R.2
  • 5
    • 9444267537 scopus 로고    scopus 로고
    • Baldwin, J., E., Williams, R., M., Eds.; Pergamon: Oxford, GB
    • (e) Clayden, J. Organolithium: Selectivity for Synthesis; Baldwin, J., E., Williams, R., M., Eds.; Pergamon: Oxford, GB, 2002; Vol. 23, pp 28-109.
    • (2002) Organolithium: Selectivity for Synthesis , vol.23 , pp. 28-109
    • Clayden, J.1
  • 18
    • 0001318042 scopus 로고    scopus 로고
    • (a) Satoh, T. Chem. Rev. 1996, 96, 3303-3326.
    • (1996) Chem. Rev. , vol.96 , pp. 3303-3326
    • Satoh, T.1
  • 34
    • 33645601418 scopus 로고    scopus 로고
    • note
    • Addition of a ligand such as TMEDA (up to 3.0 equiv) has no effect on the final result.
  • 45
    • 33645601945 scopus 로고    scopus 로고
    • note
    • Relative configuration to aminomethylphthalans 5c and 5e could be assigned on the basis of two-dimensional NOESY correlations. In the case of the cis isomers, NOE interactions between the two benzylic-type protons on C1 and C3 were diagnostic of a proximity relationship.
  • 47
    • 0030907093 scopus 로고    scopus 로고
    • For some recent reviews on the synthesis of aziridines and their reactions, see: (a) Osborn, H. M. I.; Sweeney, J. Tetrahedron: Asymmetry 1997, 8, 1693-1715.
    • (1997) Tetrahedron: Asymmetry , vol.8 , pp. 1693-1715
    • Osborn, H.M.I.1    Sweeney, J.2
  • 49
    • 1542375289 scopus 로고    scopus 로고
    • (c) Hu, X. E. Tetrahedron 2004, 60, 2701-2743.
    • (2004) Tetrahedron , vol.60 , pp. 2701-2743
    • Hu, X.E.1
  • 50
    • 0023073477 scopus 로고
    • For some recent syntheses of phthalans and phthalides, their pharmacological activity, and their uselfulness as intermediates in obtaining other bioactive compounds, see: (a) DeBernardis, J. F.; Arendsen, D. L.; Kyncl, J. J.; Kerkman, D. J. J. Med. Chem. 1987, 30, 178-184.
    • (1987) J. Med. Chem. , vol.30 , pp. 178-184
    • DeBernardis, J.F.1    Arendsen, D.L.2    Kyncl, J.J.3    Kerkman, D.J.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.