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Volumn 40, Issue 33, 1999, Pages 6101-6104

Synthesis of oxazolinyl aziridines

Author keywords

Aziridinyllithiums; Lithiation; Oxazolinyl Aziridines

Indexed keywords

AZIRIDINE DERIVATIVE; OXAZOLINE DERIVATIVE; OXAZOLINYLAZIRIDINE; UNCLASSIFIED DRUG;

EID: 0033551758     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(99)01212-5     Document Type: Article
Times cited : (32)

References (32)
  • 3
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    • For a useful review
    • For a useful review see: Tanner D. Angew. Chem. Int. Ed. Engl. 1994; 33: 599-619.
    • (1994) Chem. Int. Ed. Engl. , vol.33 , pp. 599-619
    • Angew, T.D.1
  • 9
    • 0001318042 scopus 로고    scopus 로고
    • Satoh T. Chem. Rev. 1996;96: 3303-3325 .
    • (1996) Chem. Rev. , vol.96 , pp. 3303-3325
    • Satoh, T.1
  • 10
    • 84980227255 scopus 로고
    • The deprotonation is favored by the presence of an electron-withdrawing group on the carbon of the aziridine to be deprotonated: [8a]
    • The deprotonation is favored by the presence of an electron-withdrawing group on the carbon of the aziridine to be deprotonated: [8a] Tarburton P, Chung A, Badger RC, Cromwell NH. J. Heterocyclic Chem. 1976;13: 295-300.
    • (1976) J. Heterocyclic Chem. , vol.13 , pp. 295-300
    • Tarburton, P.1    Chung, A.2    Badger, R.C.3    Cromwell, N.H.4
  • 11
    • 84980226048 scopus 로고
    • The deprotonation is favored by the presence of an electron-withdrawing group on the carbon of the aziridine to be deprotonated: [8a]
    • Tarburton P, Wall DK, Cromwell NH. ibid. 1976; 13: 411-413.
    • (1976) J. Heterocyclic Chem. , vol.13 , pp. 411-413
    • Tarburton, P.1    Wall, D.K.2    Cromwell, N.H.3
  • 24
    • 0000222273 scopus 로고
    • t-BuOCl could be conveniently prepared as described in
    • t-BuOCl could be conveniently prepared as described in: Mintz MJ, Walling C. Org. Synth., Collect. Vol. 5 1973:184-187.
    • (1973) Org. Synth., Collect. , vol.5 , pp. 184-187
    • Mintz, M.J.1    Walling, C.2
  • 26
    • 0009607645 scopus 로고    scopus 로고
    • note
    • Compound 6a could be prepared also by a Darzens-like reaction from 1b and imine 2b (60 % yield).
  • 27
    • 0009644878 scopus 로고    scopus 로고
    • note
    • 2 (390.52): calcd. C 76.89, H 7.74, N 7.17; found C 76.48, H 7.39, N 7.07.
  • 30
    • 0001449812 scopus 로고
    • 3 on the adjacent ring carbon as discussed in
    • 3 on the adjacent ring carbon as discussed in: Kingsbury CA, Durham DL, Hutton R. J. Org. Chem. 1978;43:4696-4700.
    • (1978) J. Org. Chem. , vol.43 , pp. 4696-4700
    • Kingsbury, C.A.1    Durham, D.L.2    Hutton, R.3
  • 31
    • 0001620095 scopus 로고
    • 3): δ = 0.84 (s, 3 H), 0.96 (s, 3 H), 1.53 (s, 3 H), 1.55 (s, 3 H), 3.44 (d, J = 8.0 Hz, 1 H), 3.60 (d, J = 8.0 Hz, 1 H), 6.86-7.01 (m, 3 H), 7.21-7.33 (m, 5 H), 7.48-7.53 (m, 2 H)
    • +, 445), 305 (22), 289 (1000), 247 (187), 232 (207), 144 (78), 77 (113).
    • (1970) Bull. Soc. Chim. France , vol.8-9 , pp. 3003-3010
    • Alvernhe, G.1    Laurent, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.