Carbonic anhydrase inhibitors: Inhibition of the tumor-associated isozymes IX and XII with polyfluorinated aromatic/heterocyclic sulfonamides

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 20, Issue 3, 2005, Pages 211-217

  Pastorekova, Silvia ^a   Vullo, Daniela ^b   Casini, Angela ^b   Scozzafava, Andrea ^b   Pastorek, Jaromir ^d   Nishimori, Isao ^c   Supuran, Claudiu T ^b  

^a INSTITUTE OF VIROLOGY   (Slovakia)

^b UNIVERSITY OF FLORENCE   (Italy)

^c KOCHI MEDICAL SCHOOL   (Japan)

^d NONE

Author keywords

Antitumor drug; Carbonic anhydrase; Inhibitors; Isozymes IX and XII; Polyfluorinated derivative; Sulfonamide

Indexed keywords

ACETAZOLAMIDE; ANTINEOPLASTIC AGENT; AROMATIC COMPOUND; BRINZOLAMIDE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE INHIBITOR; DICLOFENAMIDE; DORZOLAMIDE; ETHOXZOLAMIDE; HETEROCYCLIC COMPOUND; ISOENZYME; METHAZOLAMIDE; SULFONAMIDE;

ACIDIFICATION; ANTINEOPLASTIC ACTIVITY; ARTICLE; CARCINOGENESIS; CONTROLLED STUDY; CORRELATION ANALYSIS; DRUG MECHANISM; DRUG STRUCTURE; ENZYME ACTIVE SITE; ENZYME INHIBITION; GLAUCOMA; HUMAN; NONHUMAN; OUTCOMES RESEARCH; PRIORITY JOURNAL; PROGNOSIS; STRUCTURE ANALYSIS;

ANTIGENS, NEOPLASM; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; CATALYTIC DOMAIN; CLONING, MOLECULAR; ENZYME INHIBITORS; FLUOROCARBON POLYMERS; HETEROCYCLIC COMPOUNDS; HUMANS; ISOENZYMES; KINETICS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 22544439682     PISSN: 14756366     EISSN: None     Source Type: Journal    
DOI: 10.1080/14756360400028101     Document Type: Article

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