The structural basis of androgen receptor activation: Intramolecular and intermolecular amino-carboxy interactions

Proceedings of the National Academy of Sciences of the United States of America

Volumn 102, Issue 28, 2005, Pages 9802-9807

  Schaufele, Fred ^a   Carbonell, Xavier ^b   Guerbadot, Martin ^a   Borngraeber, Sabine ^a   Chapman, Mark S ^c   Ma, Aye Aye K ^b   Miner, Jeffrey N ^c   Diamond, Marc I ^b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

^c LIGAND PHARMACEUTICALS INC   (United States)

Author keywords

Conformation change; Estrogen receptor; FQNLF; FRET; Nuclear receptor

Indexed keywords

ANDROGEN RECEPTOR; ESTROGEN RECEPTOR ALPHA; HYDROXYFLUTAMIDE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA;

AMINO TERMINAL SEQUENCE; ARTICLE; CARBOXY TERMINAL SEQUENCE; CELL NUCLEUS; CONFORMATIONAL TRANSITION; CYTOPLASM; FLUORESCENCE RESONANCE ENERGY TRANSFER; HELA CELL; HORMONE RECEPTOR INTERACTION; HUMAN; HUMAN CELL; LIGAND BINDING; MOLECULAR INTERACTION; PRIORITY JOURNAL; PROTEIN FOLDING; PROTEIN PROTEIN INTERACTION; SIGNAL TRANSDUCTION;

AMINO ACID MOTIFS; BLOTTING, WESTERN; ESTROGEN RECEPTOR ALPHA; FLUORESCENCE RESONANCE ENERGY TRANSFER; FLUTAMIDE; GENETIC VECTORS; HELA CELLS; HUMANS; LIGANDS; LUCIFERASES; LUMINESCENT PROTEINS; MAMMARY TUMOR VIRUS, MOUSE; MUTATION; PPAR GAMMA; PROTEIN FOLDING; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, ANDROGEN; TRANS-ACTIVATION (GENETICS);

EID: 22244455430     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.0408819102     Document Type: Article

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