Interaction of chiral MS-245 analogs at h5-HT6 receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 15, 2005, Pages 3510-3513

  Abate, Carmen ^a   Kolanos, Renata ^a   Dukat, Malgorzata ^a   Setola, Vince ^b   Roth, Bryan L ^b,c   Glennon, Richard A ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

^b CASE WESTERN RESERVE UNIVERSITY   (United States)

^c CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Pyrrolidinylmethylindoles; Serotonin

Indexed keywords

1 BENZENESULFONYL 5 METHOXY N,N DIMETHYLTRYPTAMINE; PYRROLIDINE DERIVATIVE; SEROTONIN 6 RECEPTOR; SEROTONIN ANTAGONIST; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CHIRALITY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STRUCTURE; ENANTIOMER; ISOMER; OPTICAL ROTATION;

BINDING SITES; DRUG INTERACTIONS; HUMANS; INDOLES; PYRROLIDINES; RECEPTORS, SEROTONIN; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP; TRYPTAMINES;

EID: 21744459527     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.05.092     Document Type: Article

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