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Volumn 12, Issue 10, 2004, Pages 2797-2805

3D-QSAR CoMFA/CoMSIA studies on Urokinase plasminogen activator (uPA) inhibitors: A strategic design in novel anticancer agents

(2) Bhongade, B A a Gadad, A K a

a JAWAHARLAL NEHRU MEDICAL COLLEGE (India)

Author keywords

3D QSAR; Anticancer agents; CoMFA; CoMSIA; Indole benzoimidazole 5 carboxamidines; Urokinase plasminogen activator inhibitors

Indexed keywords

AMIDINE; ANTINEOPLASTIC AGENT; INDOLE DERIVATIVE; PLASMINOGEN ACTIVATOR INHIBITOR;

ARTICLE; COMPARATIVE MOLECULAR FIELD ANALYSIS; COMPARATIVE MOLECULAR SIMILARITY INDICES ANALYSIS; DRUG ACTIVITY; DRUG DESIGN; DRUG SELECTIVITY; DRUG STRUCTURE; HYDROGEN BOND; HYDROPHOBICITY; LIPOPHILICITY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STATISTICAL SIGNIFICANCE; STEREOSPECIFICITY; VALIDATION PROCESS;

AMIDINES; ANTINEOPLASTIC AGENTS; BENZIMIDAZOLES; DRUG DESIGN; INDOLES; MOLECULAR CONFORMATION; PLASMINOGEN INACTIVATORS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; URINARY PLASMINOGEN ACTIVATOR;

EID: 2142652097 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2004.02.019 Document Type: Article

Times cited : (30)

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