Identification of novel inhibitors of urokinase via NMR-based screening

Journal of Medicinal Chemistry

Volumn 43, Issue 21, 2000, Pages 3862-3866

  Hajduk, P J ^a   Boyd, S ^a   Nettesheim, D ^a   Nienaber, V ^a   Severin, J ^a   Smith, R ^a   Davidson, D ^a   Rockway, T ^a   Fesik, S W ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

PLASMINOGEN ACTIVATOR INHIBITOR;

ARTICLE; CHEMICAL ANALYSIS; DRUG STRUCTURE; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; STRUCTURE ANALYSIS;

BENZIMIDAZOLES; CRYSTALLOGRAPHY, X-RAY; ENZYME INHIBITORS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; STRUCTURE-ACTIVITY RELATIONSHIP; URINARY PLASMINOGEN ACTIVATOR;

EID: 0034687240     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0002228     Document Type: Article

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