Non-peptidic αvβ3 antagonists containing indol-1-yl propionic acids

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 10, 2005, Pages 2679-2684

  Leonard, Kristi ^a   Pan, Wenxi ^a   Anaclerio, Beth ^a   Gushue, Joan M ^a   Guo, Zihong ^a   DesJarlais, Renee L ^a   Chaikin, Marge A ^a   Lattanze, Jennifer ^a   Crysler, Carl ^a   Manthey, Carl L ^a   Tomczuk, Bruce E ^a   Marugan, Juan Jose ^a  

^a JOHNSON AND JOHNSON PHARMACEUTICAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

Integrins; RGD mimetic; v 3 antagonists

Indexed keywords

INDOLE DERIVATIVE; PROPIONIC ACID DERIVATIVE; VITRONECTIN RECEPTOR;

ARTICLE; CARBOXY TERMINAL SEQUENCE; DRUG POTENCY; DRUG SYNTHESIS; INHIBITION KINETICS; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

EID: 20944440970     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.01.028     Document Type: Article

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