Probing the potential of platinum(II) complexes for the inhibition of thiol-dependent enzymatic activity

Journal of Inorganic Biochemistry

Volumn 99, Issue 6, 2005, Pages 1384-1389

  Van Zutphen, Steven ^a   Kraus, Marianne ^b   Driessen, Christoph ^b   Van Der Marel, Gijs A ^a   Overkleeft, Herman S ^a   Reedijk, Jan ^a  

^a LEIDEN UNIVERSITY   (Netherlands)

^b UNIVERSITY HOSPITAL TÜBINGEN   (Germany)

Author keywords

Cathepsin; Cisplatin; Inhibitor; Platinum; Thiol dependent enzymatic activity

Indexed keywords

AMINE; CATHEPSIN B; CYSTEINE PROTEINASE; LIGAND; PLATINUM DERIVATIVE; THIOL;

ANALYTIC METHOD; ARTICLE; COMPLEX FORMATION; ENZYME ACTIVITY; ENZYME INHIBITION; EVALUATION; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

CATHEPSIN B; CYSTEINE PROTEINASE INHIBITORS; HUMANS; KINETICS; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; ORGANOPLATINUM COMPOUNDS;

EID: 19444373910     PISSN: 01620134     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jinorgbio.2005.03.014     Document Type: Article

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