Solid-water interaction. I. Study of water-pharmaceuticals interactions;Interacción sólido-agua. I. Estudio de las interacciones del agua con los sólidos farmacéuticos

Ciencia y Tecnologia Pharmaceutica

Volumn 14, Issue 1, 2004, Pages 3-12

  Bravo Osuna, I ^a   Ferrero Rodriguez C ^a   Leon Wasmer, M J ^a   Jimenez Castellanos Ballesteros, M R ^a  

^a UNIVERSITY OF SEVILLE   (Spain)

Author keywords

Absorption; Adsorption; Chemical methods; Microscopic methods; Spectroscopic methods; Thermal methods; Water amorphous solid interactions; Water crystalline solid interactions

Indexed keywords

DRUG VEHICLE; EXCIPIENT; WATER;

ADSORPTION; CHEMICAL ANALYSIS; CRYSTAL STRUCTURE; DRUG INTERACTION; HYDRATION; HYDROPHOBICITY; PHARMACEUTICS; QUALITATIVE ANALYSIS; QUANTITATIVE ANALYSIS; REVIEW; SOLID; SOLID WATER INTERACTION; SPECTROSCOPY; STOICHIOMETRY; SURFACE PROPERTY; THERMAL ANALYSIS;

EID: 1842761464     PISSN: 15753409     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review

References (44)

1. Zografi G: States of water associated with solids. Drug Dev Ind Pharm 1988; 14(14):1905-26.
2. Ford JL: Thermal analysis of hydroxypropylmethylcellulose and methylcellulose: powders, gels and matrix tablets. Int J Pharm 1999; 179:209-28.
3. Hatakeyama H, Hatakeyama T: Interaction between water and hydrophilic polymer. Therm Acta 1998; 308:3-22.
4. Roorda W: Do hydrogels contain different classes of water? J Biomater Sc Polym Edns 1994; 5:383-95.
5. Brittain HG, Bugay DE, Bogdanowich SJ y cols.: Spectral methods for determination of water. Drug Dev Ind Pharm 1988; 14(14):2029-46.
6. Clydesdale G, Roberts KJ, Telfer GB y cols.: Modeling the crystal morphology of alpha lactose monohydrate. J Pharm Sci 1997; 86:135-41.
7. Hancock B, Shamblin SL: Water vapour sorption by pharmaceutical sugars. PSTT 1998; 1(8):345-51.
8. Saleki-Gerhardt A, Stowell JG, Byrn SR y cols.: Hydratation and deshydratation of crystalline and amorphous formes of raffinose. J Pharm Sci 1995; 84:318-23.
9. Hogan SE, Buckton G: Water sorption/desorption-near IR and calorimetric study of crystalline and amorphous raffinose. Int J Pharm 2001; 227:57-69.
10. Hancock BC, Zografi G: The use of Solution Theories for predicting water vapor adsorption by amorphous pharmaceutical solids: A test of the Flory-Huggins and Vrentas Models. Pharm Res 1993; 10(9):1262-67.
11. Zografi G, Hancock BC: Water-solid state interaction in pharmaceutical systems. En Crommelin DJA, Midha K, Nagai T (Eds) Topics in Pharmaceutical Sciences Intern Pharm Federation Medpharm Scientific Publishers 1994; Stuttgart, Alemania, 415-18.
12. Thiel PA, Madey TE: The interaction of water with solid surface. Fundamental aspects. Surf Sci Rep 1987; 7:211-385.
13. Hancock BC, Zografi G: Effect of solid-state processing on water vapour sorption by aspirin. J Pharm Sci 1996; 85:246-8.
14. Jakobsen DF, Frokjaer S, Larsen C y cols.: Application of isothermal microcalorimetry in preformulation I. Hygroscopicity of drug substances Int J Pharm 1997; 156: 67-77.
15. Down GRB, Mc Mullen JN: The effect of interparticulate friction and moisture on the crushing strength of sodium chloride compacts. Powder Tech 1985; 42:169.
16. Bauer J, Quick J, Oheim R: Alternative interpretation of the role of water in the erytromycin structure. J Pharm Sci 1985; 74:899-900.
17. Pande GS, Shangraw RF: Characterization of (-cyclodextrin of direct compression tableting. The role of moisture in the compactibility of β-cyclodextrin. Int J Pharm 1995; 124:231-9.
18. Suihko E, Ketolainen J, Poso A y cols.: Dehydratation of theophylline monohydrate- A two step process. Int J Pharm 1997; 158:47-55.
19. Dawoodbhai S, Rhodes CT: The effect of moisture on powder flow and on compactation and physical stability of tablets. Drug Dev Ind Pharm 1989; 15(10):1577-600
20. Stubberud I, Arwidsson HG, Larsson A y cols.: Water solid interactions II. Effect of moisture sorption and glass transition temperature on compactability of microcrystalline cellulose alone or in binary mixture with polyvinil pyrrolidone. Int J Pharm 1996; 134:79-88.
21. Faroongsarng D, Peck GE: The swelling and water uptake of tablets. III: moisture sorption behavior of tablet disintegrants. Drug Dev Ind Pharm 1994; 20(5):779-98.
22. Maa YF, Nguyen PA, Andya JD y cols.: Effect of spray drying and subsequent processing conditions on residual moisture content and physical/biochemical stability of protein inhalation powders. Pharm Res 1998; 15(5):768-75.
23. Sebhatu T, Elamin AA, Ahlneck C: Effect of moisture sorption on tabletting characteristics of spray dried (15% amorphous) lactose. Pharm Res 1994; 11(9):1233-8.
24. Mathlouthi M: Water content, water activity, water structure and the stability of foodtuffs. Food Control 2001; 12:409-17.
25. Dalton CR, Hancock BC: Proc;essing and storage effects on water vapor sorption by some model pharmaceutical solid dosage formulations. Int J Pharm 1997; 156:143-51.
26. Hollenbeck RG: Moisture in Pharmaceutical products En Encyclopedia of Pharmaceutical Technology. Swarbrick J, Boyland JC (Eds), Marcel Dekker, INC. New York 1988; 10
27. Troller JA, Christian JHB: Water activity and food, New York Academic Press. New York 1978: 13-47.
28. Vornhof DW, Thomas JH: Determination of moisture in starch hydrolisates by near-infrared and infrared spectrophotometry. Anal Chem 1970; 42:1230.
29. Isegard, HD: Rapid water determination in foodstuffs. Trends Food Sci Techn 1995; 6:155-62
30. Marshall K, Sixsmith D: Some physical characteristics of microcrystalline cellulose powders. Drug Dev Ind Comm 1975; 1:51-7.
31. 13C CP-MAS NMR spectroscopy I: Spectral decomposition. Carbohydr Polym 1999; 39:327-39.
32. Hopkinson I, Jones RAL, McDonald PJ y cols.: Water ingress into starch and sucrose:starch systems. Polymer 2001; 4:4947-56.
33. Ford JL, Timmins P: Pharmaceutical thermal analysis Techniques and applications. Ellis Horwood limited, Chichester, West Sussex, England 1989.
34. Coleman NJ, Craig DQM: Modulated temperature differential scanning calorimetry: a novel approach to pharmaceutical thermal analysis. Int J Pharm 1996; 135:13-29.
35. Hatakeyama T, Quinn FX: Thermal analysis Fundamentals and applications to polymer science, 2nd edition. (Eds) John Wiley and sons (Eds), Chichester, West Sussex, England 1999.
36. Clas SD, Dalton CR, Hancock BC: Differential scanning calorimetry: applications in drug development. PSTT 1999; 2(8):311-20.
37. Kerc J, Srcic S, Mohar M y cols.: Some physicochemical properties of glassy felodipine. Int J Pharm 1991; 68:25-33.
38. Steendam R, Frijlink WH, Lerk CF: Plastification of amylodextrin by moisture. Consecuences for compaction behaviour and tablets properties. Eur J Pharm Sci 2001; 14:245-54
39. van der Voort Maarschalk K, Vromans H, Bolhuis GK y cols.: Influence of plasticizers on tableting properties of polymers. Drug Dev Ind Pharm 1998; 24(3):261-68.
40. Steendam R, Eissens ACE; Frijlink WH y cols.: Plastification of amylodextrin by moisture. Consecuences for drug release from tablets. Int J Pharm 2000; 20:23-33.
41. Gordon M, Taylor JS: Ideal copolymers and second order transition of synthetic rubbers. 1. Non-crystalline copolymers. J Appl Chem 1952; 2:493-500.
42. Price DM, Reading M, Hammiche A y cols.: Microthermal analysis: scanning thermal microscopy and localised thermal analysis. Int J Pharm 1999; 192:85-96.
43. Bravo-Osuna I, Muñoz-Ruiz A, Jiménez-Castellanos MR y cols.: Aspects of sample encapsulation on the apparent glass transition and other transitions of methylmethacrylate copolymers measured by MTDSC and DSC. J Therm Anal Calorim 2002; 69:387-407.
44. Badawy SIF, Gawronski AJ, Alvarez FJ: Application of sorption-desorption moisture transfer modeling to the study of chemical stability of a moisture sensitive drug product in different packaging configurations. Int J Pharm 2001; 223:1-13.