N,N-Dialkyl-4-[(8-azabicyclo[3.2.1]-oct-3-ylidene)phenylmethyl]benzamides, potent, selective δ opioid agonists

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 9, 2004, Pages 2109-2112

  Carson, John R ^a   Coats, Steven J ^a   Codd, Ellen E ^a   Dax, Scott L ^a   Lee, Jung ^a   Martinez, Rebecca P ^a   Neilson, Lou Anne ^a,b   Pitis, Philip M ^a   Zhang, Sui Po ^a  

^a JOHNSON AND JOHNSON PHARMACEUTICAL RESEARCH AND DEVELOPMENT   (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZAMIDE DERIVATIVE; DELTA OPIATE RECEPTOR; DELTA OPIATE RECEPTOR AGONIST; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); MU OPIATE RECEPTOR;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTINOCICEPTION; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; MOUSE; NONHUMAN; STIMULATION;

ANALGESICS, OPIOID; BENZAMIDES; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); RECEPTORS, OPIOID, DELTA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 1842690631     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.02.051     Document Type: Article

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