In vitro and in vivo activity of analogues of the kinin B2 receptor antagonist men112701

Canadian Journal of Physiology and Pharmacology

Volumn 80, Issue 4, 2002, Pages 293-302

  Meini, S ^a   Lecci, A ^a   Carini, F ^a   Tramontana, M ^a   Giuliani, S ^a   Maggi, C A ^a   Ricci, R ^a   Fabbri, G ^a   Anichini, B ^a   Harmat, N ^a   Rizzi, A ^a   Camarda, V ^a   Regoli, D ^a   Quartara, L ^a  

^a Pharmacology Department   (Italy)

Author keywords

Asthma; Blood pressure; Bradykinin; Guinea pig; Metabolism

Indexed keywords

AMINOPEPTIDASE; BRADYKININ; BRADYKININ B2 RECEPTOR ANTAGONIST; DIPEPTIDYL CARBOXYPEPTIDASE; MEN 11270; MEN 12374; MEN 12388; MEN 12739; MEN 13031; MEN 13052; MEN 13346; MEN 13371; MEN 13405; MEN 13655; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; BINDING AFFINITY; BRONCHOSPASM; CHO CELL; CONCENTRATION RESPONSE; CONFERENCE PAPER; CONTROLLED STUDY; DRUG ACTIVITY; DRUG ANTAGONISM; DRUG DEGRADATION; DRUG EFFECT; DRUG POTENCY; DRUG RECEPTOR BINDING; ENZYME DEGRADATION; FEMALE; GUINEA PIG; HUMAN; HUMAN TISSUE; HYPOTENSION; ILEUM; ILEUM CONTRACTION; IN VITRO STUDY; IN VIVO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN LOCALIZATION; UMBILICAL VEIN; VENOCONSTRICTION;

ADULT; ANIMALS; BRADYKININ; BRONCHOCONSTRICTION; CHO CELLS; CRICETINAE; FEMALE; GUINEA PIGS; HUMANS; HYPOTENSION; INJECTIONS, INTRAVENOUS; MALE; OLIGOPEPTIDES; PEPTIDES, CYCLIC; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ;

EID: 18344394948     PISSN: 00084212     EISSN: None     Source Type: Journal    
DOI: 10.1139/y02-022     Document Type: Conference Paper

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