Receptors for kinins in the human isolated umbilical vein

British Journal of Pharmacology

Volumn 118, Issue 2, 1996, Pages 289-294

  Gobeil, F ^a   Pheng, L H ^a   Badini, I ^a   Nguyen Le, X K ^a   Pizard, A ^a   Rizzi, A ^a   Blouin, D ^b   Regoli, D ^a  

^a UNIVERSITÉ DE SHERBROOKE   (Canada)

^b CENTRE HOSPITALIER UNIVERSITAIRE DE SHERBROOKE   (Canada)

Author keywords

Agonists; Antagonists; B1 and B2 receptors; Bradykinin; Human umbilical vein; Smooth muscle

Indexed keywords

BRADYKININ; BRADYKININ ANTAGONIST; BRADYKININ B1 RECEPTOR; BRADYKININ B2 RECEPTOR; BRADYKININ DERIVATIVE; BRADYKININ RECEPTOR AGONIST; BRADYKININ[8 LEUCINE 9 DEARGININE]; ICATIBANT; [[4 [2 [[BIS(CYCLOHEXYLAMINO)METHYLENE]AMINO] 3 (2 NAPHTHYL)PROPIONAMIDO]PHENYL]METHYL]TRIBUTYLPHOSPHONIUM CHLORIDE;

ADULT; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; FEMALE; HUMAN; HUMAN TISSUE; NORMAL HUMAN; PRIORITY JOURNAL; UMBILICAL VEIN; VENOCONSTRICTION;

EID: 0030010048     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1476-5381.1996.tb15401.x     Document Type: Article

References (28)

1. ALTURA, B.M., MALAVIYA, D., REICH, F.C. & ORKIN, L.R. (1972). Effects of vasoactive agents on isolated human umbilical arteries and veins. Am. J. Physiol., 222, 354-355.
2. COUTURE, R., MIZRAHI, J., REGOLI, D. & DEVROEDE, G. (1981). Peptides and the human colon: an in vitro pharmacological study. Can. J. Physiol. Pharmacol., 59, 957-964.
3. DRAPEAU, G. & REGOLI, D. (1988). Synthesis of bradykinin analogs. Methods Enzymol., 163, 263-272.
4. 2 receptor gene. Biochem. Biophys. Res. Commun., 187, 1306-1313.
5. FÉLÉTOU, M., MARTIN, C.A.E., MOLIMARD, M., NALINE, E., GERMAIN, M., THURIAU, C., FAUCHÈRE, J-L., CANET, E. & ADVENIER, C. (1995). In vitro effects of HOE 140 in human bronchial and vascular tissue. Eur. J. Pharmacol., 274, 57-64.
6. GOBEIL, F. & REGOLI, D. (1994). Characterization of kinin receptors by bioassays. Braz. J. Med. Biol. Res., 27, 1781-1791.
7. 9-Bradykinin. J. Biol. Chem., 259, 9263-9268.
8. 2 bradykinin receptors. Mol. Pharmacol., 45, 1-8.
9. HESS, J.F., BORKOWSKI, H.A., YOUNG, G.S., STRADER, C.D. & RANSOM, R.W. (1992). Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor. Biochem. Biophys. Res. Commun., 184, 260-268.
10. HOCK, F.J., WIRTH, K., ALBUS, U., LINZ, W., GERHARDS, H.J., WIEMER, G., HENKE, ST., BREIPOHL, G., KÖNIG, W., KNOLLE, J. & SCHÖLKENS, B.A. (1991). Hoe 140, a new potent and long acting bradykinin-antagonist: in vitro studies. Br. J. Pharmacol., 102, 769-773.
11. 1 receptors: a review. Immunopharmacology, 30, 1-26.
12. 2 receptors on the venoconstrictor action of bradykinin. J. Pharmacol. Exp. Ther., 269, 1136-1143.
13. 2 bradykinin receptor. Proc. Natl. Acad. Sci. U.S.A., 88, 7724-7728.
14. 1 receptor. Biochim. Biophys. Acta., 1264, 223-228.
15. MENKE, J.G., BORKOWSKI, J.A., BIERILO, K.K., MCNEIL, T., DERRICK, A.W., SCHNECK, K.A., RAMSON, R.W., STRADER, C.D., LINESNEYER, D.L. & HESS, J.F. (1994). Expression cloning of a human B-1 bradykinin receptor. J. Biol. Chem., 269, 21583-21586.
16. REGOLI, D. & BARABÉ, J. (1980). Pharmacology of bradykinin and related kinins. Pharmacol. Rev., 32, 1-46.
17. REGOLI, D., BARABÉ, J. & PARK, W.K. (1977). Receptors of bradykinin in rabbit aorta. Can. J. Physiol. Pharmacol., 55, 855-867.
18. REGOLI, D., BOUDON, A. & FAUCHÈRE, J.L. (1994a). Receptors and antagonists for substance P and related peptides. Pharmacol. Rev., 46, 551-599.
19. 2 subtypes. Life Sci., 55, 735-749.
20. REGOLI, D., JUKIC, D., GOBEIL, F. & RHALEB, N.-E. (1993). Receptors for bradykinin and related kinins: a critical analysis. Can. J. Physiol. Pharmacol., 71, 556-567.
21. 2 receptor characterization. Trends Pharmacol. Sci., 11, 156-161.
22. RHALEB, N.-E., DRAPEAU, G., DION, S., JUKIC, D., ROUISSI, N. & REGOLI, D. (1990). Structure-activity studies on bradykinin and related peptides. Agonists. Br. J. Pharmacol., 99, 445-448.
23. 2 receptor antagonists. Hypertension, 17, 107-115.
24. 2 receptor. J. Med. Chem., 36, 2583-2584.
25. SCHILD, H.O. (1947). pA, a new scale for the measurement of drug antagonism. Br. J. Pharmacol. Chemother., 2, 189-202.
26. SCHILD, H.O. (1973). Receptor classification with special reference to beta adrenergic receptors. In Drug Receptors, pp. 29-36. ed. Rang, H.P. Baltimore, U.S.A.: University Park Press.
27. nd ed.), New York, U.S.A.: Springer Verlag.
28. WIRTH, K., HOCK, F.J., ALBUS, U., LINZ, W., ALPERMANN, H.G., ANAGNOSTOPULOS, H., HENKE, S., BREIPOHE, G , KÖNIG, W., KNOLLE, J. & SCHÖLKENS, B.A. (1991). Hoe 140 a new potent and low acting bradykinin antagonist. Br. J. Pharmacol., 102, 774-777.