Peptide and non-peptide bradykinin B2 receptor agonists and antagonists: A reappraisal of their pharmacology in the guinea-pig ileum

European Journal of Pharmacology

Volumn 409, Issue 2, 2000, Pages 185-194

  Meini, Stefania ^a   Patacchini, Riccardo ^a   Lecci, Alessandro ^a   Quartara, Laura ^a   Maggi, Carlo Alberto ^a  

^a Menarini Ricerche SpA   (Italy)

Author keywords

Antagonism; Bradykinin B2 receptor; FR173657; FR190997; MEN 11270; Non peptide

Indexed keywords

3 (6 ACETAMIDO 3 PYRIDYL) N [N [2,4 DICHLORO 3 [(2 METHYL 8 QUINOLINYL)OXYMETHYL]PHENYL] N METHYLAMINOCARBONYLMETHYL]ACRYLAMIDE; 8 [2,6 DICHLORO 3 [N [4 (N METHYLCARBAMOYL)CINNAMAMIDOACETYL] N METHYLAMINO]BENZYLOXY] 2 METHYL 4 (2 PYRIDYLMETHOXY)QUINOLINE; 8 [2,6 DICHLORO 3 [N [4(N METHYLCARBAMOYL)CINNAMIDOACETYL] N METHYLAMINO]BENZYLOXY] 2 METHYL 4 (2 PYRIDYLMETHOXY)QUINOLINE; BRADYKININ; BRADYKININ B2 RECEPTOR; BRADYKININ B2 RECEPTOR AGONIST; BRADYKININ B2 RECEPTOR ANTAGONIST; ICATIBANT; MEN 11270; PARTIAL AGONIST; PEPTIDE; TRITIUM; UNCLASSIFIED DRUG;

AGONIST; ANIMAL TISSUE; ARTICLE; BINDING COMPETITION; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG RECEPTOR BINDING; GUINEA PIG; ILEUM; MALE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; SMOOTH MUSCLE CONTRACTILITY;

ANIMALS; BINDING, COMPETITIVE; BRADYKININ; DOSE-RESPONSE RELATIONSHIP, DRUG; GUINEA PIGS; ILEUM; MALE; MEMBRANES; MUSCLE CONTRACTION; MUSCLE, SMOOTH; OLIGOPEPTIDES; PEPTIDES, CYCLIC; QUINOLINES; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ;

EID: 0034624258     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(00)00850-5     Document Type: Article

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