Differences between peptide and nonpeptide B2 bradykinin receptor antagonists in blocking bronchoconstriction and hypotension induced by bradykinin in anesthetized guinea pigs

Journal of Pharmacology and Experimental Therapeutics

Volumn 296, Issue 3, 2001, Pages 1051-1057

  Tramontana, Manuela ^a   Lecci, Alessandro ^a   Meini, Stefania ^a   Montserrat, Xavier ^b   Pascual, Jaume ^b   Giuliani, Sandro ^a   Quartara, Laura ^a   Maggi, Carlo Alberto ^a  

^a Menarini Ricerche SpA   (Italy)

^b Laboratorios Menarini   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

3 (6 ACETAMIDO 3 PYRIDYL) N [N [2,4 DICHLORO 3 [(2 METHYL 8 QUINOLINYL)OXYMETHYL]PHENYL] N METHYLAMINOCARBONYLMETHYL]ACRYLAMIDE; BRADYKININ; BRADYKININ B2 RECEPTOR ANTAGONIST; ICATIBANT; MEN 11270; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BRONCHOSPASM; CONTROLLED STUDY; DRUG EFFECT; DRUG EFFICACY; DRUG METABOLISM; DRUG STABILITY; GUINEA PIG; HYPOTENSION; MALE; NONHUMAN; PRIORITY JOURNAL;

ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; BLOOD PRESSURE; BRADYKININ; BRONCHOCONSTRICTION; CELL MEMBRANE; DISEASE MODELS, ANIMAL; DRUG INTERACTIONS; DRUG STABILITY; GUINEA PIGS; HYPOTENSION; INFUSIONS, INTRAVENOUS; LUNG; MALE; OLIGOPEPTIDES; PEPTIDES, CYCLIC; QUINOLINES; RECEPTOR, BRADYKININ B2; RECEPTORS, BRADYKININ; TRITIUM;

EID: 0035119601     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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