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Volumn 10, Issue 2, 2002, Pages 361-369

Synthesis and biological activity of new 1,4-benzodioxan-arylpiperazine derivatives. Further validation of a pharmacophore model for α1-adrenoceptor antagonists

(9) Barbaro, Roberta a Betti, Laura b Botta, Maurizio c Corelli, Federico c Giannaccini, Gino b Maccari, Laura c Manetti, Fabrizio c Strappaghetti, Giovannella a Corsano, Stefano a

a UNIVERSITY OF PERUGIA (Italy)

b UNIVERSITY OF PISA (Italy)

c UNIVERSITY OF SIENA (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 BENZODIOXANARYLPIPERAZINE DERIVATIVE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; METHYL GROUP; NITROGEN; PIPERAZINE; PIPERAZINE DERIVATIVE; PRAZOSIN; PYRIDAZINONE DERIVATIVE; PYRIDINE; RADIOLIGAND; RAUWOLSCINE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; ENANTIOMER; NONHUMAN; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; DRUG EVALUATION, PRECLINICAL; MODELS, MOLECULAR; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0036132213 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00286-3 Document Type: Article

Times cited : (44)

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