2,3-bis(5-alkyl-2-thiono-1,3,5-thiadiazin-3-yl) propionic acid: One-pot Domino synthesis and antimicrobial activity

Archiv der Pharmazie

Volumn 338, Issue 1, 2005, Pages 38-43

  El Bialy, Serry A A ^a,c   Abdelal, Ali M ^a   El Shorbagi, Abdel Nasser ^b   Kheira, Samy M M ^a  

^a MANSOURA UNIVERSITY   (Egypt)

^b Assiut University   (Egypt)

^c UNIVERSITY OF TOKYO   (Japan)

Author keywords

Bis(2 thiono tetrahydro 2H 1,3,5 thiadiazine); Domino reaction, Antibacterial and antifungal activity

Indexed keywords

ALIPHATIC AMINE; ALKYL GROUP; ANTIFUNGAL AGENT; ANTIINFECTIVE AGENT; CARBON DISULFIDE; CIPROFLOXACIN; DIMETHYLAMINE; FORMALDEHYDE; NALIDIXIC ACID; PHOSPHORUS DERIVATIVE; PROPIONAMIDE DERIVATIVE; PROPIONIC ACID DERIVATIVE; THIADIAZINE DERIVATIVE;

ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ASPERGILLUS FLAVUS; BACTERIAL STRAIN; CANDIDA ALBICANS; DRUG SCREENING; DRUG SYNTHESIS; FUNGUS GROWTH; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; IN VITRO STUDY; NONHUMAN; PENICILLIUM EXPANSUM; PRIORITY JOURNAL; REACTION ANALYSIS; SPOROGENESIS; STRUCTURE ACTIVITY RELATION; TRICHODERMA HARZIANUM;

ANTI-BACTERIAL AGENTS; ANTIFUNGAL AGENTS; ASPERGILLUS FLAVUS; CANDIDA ALBICANS; GRAM-NEGATIVE BACTERIA; GRAM-POSITIVE BACTERIA; MICROBIAL SENSITIVITY TESTS; PROPIONIC ACIDS; STRUCTURE-ACTIVITY RELATIONSHIP; THIADIAZINES; THIONES; TRICHODERMA;

EID: 14944381732     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.200400906     Document Type: Article

References (33)

1. th ed., John Wiley and Sons, New York, 1979, chapter 22.
2. A. El-Shorbagi, Arch. Pharm. Pharm. Med. Chem. 2000, 333, 281-286.
3. T. Aboul-Fadl, K. Hassanin, Pharmazie 1999, 54, 244-247.
4. T. Aboul-Fadl, A. El-Shorbagi, Arch. Pharm. Pharm. Med. Chem. 1997, 330, 327-332.
5. T. Aboul-Fadl, A. El-Shorbagi, Eur. J. Med. Chem. 1996, 31, 165-169.
6. A. El-Shorbagi, Eur. J. Med. Chem. 1994, 29, 11-19.
7. M. Ertan, A. A. Bilgil, E. Palaska, N. Yulug, Arzneim-Forsch./-Drug Res. 1992, 42, 160-163.
8. M. Ertan, S. Sarac, N. Yulug, Arzneim-Forsch./Drug Res. 1990, 40, 790-765.
9. M. Ertan, A. B. Tayhan, N. Yulug, Arch. Pharm. 1990, 323, 605-609.
10. T. Zsolanai, Arzneim-Forsch./Drug Res. 1971, 21, 121-127.
11. T. Zsolanai, Arzneim-Forsch./Drug Res. 1968, 18, 1319-1324.
12. A. Reiche, G. Hilgetag, A. Martini, R. Philppson, Arch. Pharm. 1961, 294, 201-209.
13. D. T. W. Chu, P. B. Fernandes, Adv. Drug Res. 1991, 21, 39.
14. R. Cipro, O. Perez, M. Reyes, H. E. Suarez Garay, L. J. Cruz, H. Rodriguez, M. D. Molero-Vilchez, C. Ochoa, Tetrahedron Lett. 2000, 47, 613.
15. S. Muelas, M. Suarez, R. Perez, H. Rodriguez, C. Ochoa, J.A. Escario, A. Gomez-Barrio, Mem Institute Oswaldo Cruz, Rio de Janeiro, 2002, 97, 269. (International Conference)
16. C. Ochoa, E. Perez, R. Perez, M. Suarez, E. Ochoa, H. Rodriguez, A. Gomez-Barrio, S. Muelas, J. J. Nogal, R. A. Martinez, Arzneim-Forsch./Drug Res. 1999, 49, 764-769.
17. T. Aboul-Fadl, M. A. Hussein, A. El-Shorbagi, A-R Khallil, Arch. Pharm. Pharm. Med. Chem. 2002, 3354, 438-442.
18. A. M. Abdelal, S. M. Kheira, F. A. Badria, Sci. Pharm. 1997, 65, 99-106.
19. M. A. Hussein, A. El-Shorbagi, A-R Khallil, Arch. Pharm. Pharm. Med. Chem., 2001, 334, 305-308.
20. M. Tramontini, Synthesis 1973, 703-775.
21. L. F Tietze, Chem. Rev. 1996, 96, 115-136.
22. L. F. Tietze, U. Beifuss, Angew. Chem. Int. Ed. Engl. 1993, 32, 131-163.
23. L. F. Tietze, Chem. Ind. 1995, 453. H. Waldmann, in Domino Reaction in Organic Synthesisp Highlight II; (Ed.: H. Waldmann), VCH, Weinheim, 1995, pp 193-202. Hall, N., Science 1994, 266, 32-35.
24. L. F. Tietze, Chem. Ind. 1995, 453. H. Waldmann, in Domino Reaction in Organic Synthesisp Highlight II; (Ed.: H. Waldmann), VCH, Weinheim, 1995, pp 193-202. Hall, N., Science 1994, 266, 32-35.
25. L. F. Tietze, Chem. Ind. 1995, 453. H. Waldmann, in Domino Reaction in Organic Synthesisp Highlight II; (Ed.: H. Waldmann), VCH, Weinheim, 1995, pp 193-202. Hall, N., Science 1994, 266, 32-35.
26. Y. Kageyama, Y. Yamazaki, H. Okuno, J. Inorg. Biochem. 1998, 70, 25-32.
27. H. F. Kung, C. C. Yu, J. Billings, M. Blau, J. Med. Chem., 1935, 28, 1280-1284.
28. E. F. Godefoi, U.S. Patent 2738368. [Chem. Abstr. 1957, 51, 463f].
29. S.R. Jain, A. Kar, Planta Med. 1971, 20, 118-123.
30. R. Wise, T. M. Andrews, L. Edward, Antimicrob. Ag. Chemother. 1983, 23, 559-564.
31. S. T. Pai, M. W. Platt, Letter in Applied Microbiology 1995, 20, 14-18.
32. S. A. Ouf, S. M. Sherif, Folia Microbiol. 1993, 38, 181-187.
33. T. P. West, Microbios 1988, 226, 27-36.