메뉴 건너뛰기




Volumn 10, Issue 1, 2005, Pages 97-104

Effect of chemical penetration enhancer and iontophoresis on the in vitro percutaneous absorption enhancement of insulin through porcine epidermis

Author keywords

Fatty acids; Iontophoresis; Limonene; Permeability; Permeation enhancer; Transdermal

Indexed keywords

ACETIC ACID ETHYL ESTER; FATTY ACID; INSULIN LISPRO; LIMONENE; LINOLEIC ACID; LINOLENIC ACID; OLEIC ACID; PALMITIC ACID; PALMITOLEIC ACID; PROPYLENE GLYCOL; RECOMBINANT HUMAN INSULIN; STEARIC ACID;

EID: 14644395611     PISSN: 10837450     EISSN: None     Source Type: Journal    
DOI: 10.1081/PDT-200049679     Document Type: Article
Times cited : (30)

References (37)
  • 1
    • 0032883241 scopus 로고    scopus 로고
    • Transdermal penetration enhancers: Applications, limitations, and potential
    • Finnin, B.C.; Morgan, T.M. Transdermal penetration enhancers: applications, limitations, and potential. J. Pharm. Sci. 1999, 88, 955-958.
    • (1999) J. Pharm. Sci. , vol.88 , pp. 955-958
    • Finnin, B.C.1    Morgan, T.M.2
  • 4
    • 0033812031 scopus 로고    scopus 로고
    • Mechanism(s) of in vitro percutaneous absorption enhancement of tamoxifen by enhancers
    • Zhao, K.D.; Singh, J. Mechanism(s) of in vitro percutaneous absorption enhancement of tamoxifen by enhancers. J. Pharm. Sci. 2000, 89, 771-780.
    • (2000) J. Pharm. Sci. , vol.89 , pp. 771-780
    • Zhao, K.D.1    Singh, J.2
  • 5
    • 0034493157 scopus 로고    scopus 로고
    • Synergistic effect of enhancers for transdermal drug delivery
    • Mitragotri, S. Synergistic effect of enhancers for transdermal drug delivery. Pharm. Res. 2000, 17, 1354-1359.
    • (2000) Pharm. Res. , vol.17 , pp. 1354-1359
    • Mitragotri, S.1
  • 6
    • 0036079241 scopus 로고    scopus 로고
    • Effect of permeation enhancer pretreatment on the iontophoresis of luteinizing hormone releasing hormone (LHRH) through human epidermal membrane (HEM)
    • Smyth, H.D.C.; Becket, C.; Mehta, S. Effect of permeation enhancer pretreatment on the iontophoresis of luteinizing hormone releasing hormone (LHRH) through human epidermal membrane (HEM). J. Pharm. Sci. 2002, 91, 1296-1307.
    • (2002) J. Pharm. Sci. , vol.91 , pp. 1296-1307
    • Smyth, H.D.C.1    Becket, C.2    Mehta, S.3
  • 7
    • 0023597397 scopus 로고
    • Mode of action of penetration enhancers in human skin
    • Barry, B.W. Mode of action of penetration enhancers in human skin. J. Control. Release 1987, 6, 85-97.
    • (1987) J. Control. Release , vol.6 , pp. 85-97
    • Barry, B.W.1
  • 8
  • 9
    • 0002512224 scopus 로고
    • Fatty acids as skin permeation enhancers
    • Hsieh, D.S., Ed.; Marcel Dekker: Basal
    • Aungst, B.J. Fatty acids as skin permeation enhancers. In Percutaneous Penetration Enhancer; Hsieh, D.S., Ed.; Marcel Dekker: Basal, 1994; 277-285.
    • (1994) Percutaneous Penetration Enhancer , pp. 277-285
    • Aungst, B.J.1
  • 10
    • 0031926051 scopus 로고    scopus 로고
    • Synergistic effect of iontophoresis and a series of fatty acids on LHRH permeability through porcine skin
    • Bhatia, K.S.; Singh, J. Synergistic effect of iontophoresis and a series of fatty acids on LHRH permeability through porcine skin. J. Pharm. Sci. 1998, 87, 462-469.
    • (1998) J. Pharm. Sci. , vol.87 , pp. 462-469
    • Bhatia, K.S.1    Singh, J.2
  • 11
    • 0021182767 scopus 로고
    • Increased skin permeability for lipophilic molecules
    • Cooper, E.R. Increased skin permeability for lipophilic molecules. J. Pharm. Sci. 1984, 73, 1153-1156.
    • (1984) J. Pharm. Sci. , vol.73 , pp. 1153-1156
    • Cooper, E.R.1
  • 12
    • 0025102626 scopus 로고
    • Percutaneous absorption promoting effect and skin irritancy of monocyclic monoterpenes
    • Okabe, H.; Obata, Y.; Takayama, K.; Nagai, T. Percutaneous absorption promoting effect and skin irritancy of monocyclic monoterpenes. Drug. Des. Deliv. 1990, 6, 229-238.
    • (1990) Drug. Des. Deliv. , vol.6 , pp. 229-238
    • Okabe, H.1    Obata, Y.2    Takayama, K.3    Nagai, T.4
  • 14
    • 0029644942 scopus 로고
    • Role of C-terminal B-chain residues in insulin assembly; the structure of hexameric Lys B28 Pro B29-human insulin
    • Ciszak, E.; Beals, J.M.; Frank, B.H.; Baker, J.C.; Carter, N.D.; Smith, G.D. Role of C-terminal B-chain residues in insulin assembly; the structure of hexameric Lys B28 Pro B29-human insulin. Structure 1995, 3, 615-622.
    • (1995) Structure , vol.3 , pp. 615-622
    • Ciszak, E.1    Beals, J.M.2    Frank, B.H.3    Baker, J.C.4    Carter, N.D.5    Smith, G.D.6
  • 15
    • 0016373013 scopus 로고
    • Percutaneous penetration of some pesticides and herbicides in man
    • Feldman, R.J.; Maibach, H.I. Percutaneous penetration of some pesticides and herbicides in man. Toxicol. Appl. Pharmacol. 1974, 28, 126-132.
    • (1974) Toxicol. Appl. Pharmacol. , vol.28 , pp. 126-132
    • Feldman, R.J.1    Maibach, H.I.2
  • 16
    • 0000236054 scopus 로고
    • In vivo animal models for percutaneous absorption
    • Bronaugh, R.L., Maibach, H.I., Eds.; Marcel Dekker: New York
    • Wester, R.C.; Maibach, H.I. In vivo animal models for percutaneous absorption. In Percutaneous Absorption; Bronaugh, R.L., Maibach, H.I., Eds.; Marcel Dekker: New York, 1989; 221-238.
    • (1989) Percutaneous Absorption , pp. 221-238
    • Wester, R.C.1    Maibach, H.I.2
  • 17
    • 0030319632 scopus 로고    scopus 로고
    • Pig ear skin as a model for predicting percutaneous absorption in man
    • Bhatia, K.S.; Singh, J. Pig ear skin as a model for predicting percutaneous absorption in man. Pharm. Sci. 1996, 2, 275-276.
    • (1996) Pharm. Sci. , vol.2 , pp. 275-276
    • Bhatia, K.S.1    Singh, J.2
  • 18
    • 0031003156 scopus 로고    scopus 로고
    • Effect of penetration enhancers and iontophoresis in the FT-IR spectroscopy and LHRH permeability through porcine skin
    • Bhatia, K.S.; Gao, S.; Singh, J. Effect of penetration enhancers and iontophoresis in the FT-IR spectroscopy and LHRH permeability through porcine skin. J. Control. Release 1997, 47, 81-89.
    • (1997) J. Control. Release , vol.47 , pp. 81-89
    • Bhatia, K.S.1    Gao, S.2    Singh, J.3
  • 19
    • 0003115728 scopus 로고
    • Technological and developmental issues of iontophoretic transport of peptide and protein drugs
    • Lee, V.H.L., Hashida, M., Mizushima, Y., Eds.; Harwood Academic Publishers: Chur, Switzerland
    • Sage, B.H., Jr.; Bock, C.R.; Denuzzio, J.D.; Hoke, R.A. Technological and developmental issues of iontophoretic transport of peptide and protein drugs. In Trends and Future Perspectives in Peptide and Protein Drug Delivery; Lee, V.H.L., Hashida, M., Mizushima, Y., Eds.; Harwood Academic Publishers: Chur, Switzerland, 1995; 111-134.
    • (1995) Trends and Future Perspectives in Peptide and Protein Drug Delivery , pp. 111-134
    • Sage Jr., B.H.1    Bock, C.R.2    Denuzzio, J.D.3    Hoke, R.A.4
  • 20
    • 0019976664 scopus 로고
    • Correction of perfusate concentration for sample removal
    • Hayton, W.L.; Chen, T. Correction of perfusate concentration for sample removal. J. Pharm. Sci. 1982, 71, 820-821.
    • (1982) J. Pharm. Sci. , vol.71 , pp. 820-821
    • Hayton, W.L.1    Chen, T.2
  • 22
    • 0035857712 scopus 로고    scopus 로고
    • Lipid extraction and iontophoretic transport of leuprolide acetate through porcine epidermis
    • Rastogi, S.K.; Singh, J. Lipid extraction and iontophoretic transport of leuprolide acetate through porcine epidermis. Int. J. Pharm. 2001, 215, 241-249.
    • (2001) Int. J. Pharm. , vol.215 , pp. 241-249
    • Rastogi, S.K.1    Singh, J.2
  • 23
    • 0002611260 scopus 로고
    • Simple alkyl esters as skin penetration enhancers
    • Walters, K.A., Hadgraft, J., Eds.; Marcel Dekker: New York
    • Friend, D.R.; Heller, J. Simple alkyl esters as skin penetration enhancers. In Pharmaceutical Skin Penetration Enhancement; Walters, K.A., Hadgraft, J., Eds.; Marcel Dekker: New York, 1993; 31-56.
    • (1993) Pharmaceutical Skin Penetration Enhancement , pp. 31-56
    • Friend, D.R.1    Heller, J.2
  • 24
    • 0024467413 scopus 로고
    • Alkyl esters as skin permeation enhancers for indomethacin
    • Catz, P.; Friend, R.D. Alkyl esters as skin permeation enhancers for indomethacin. Int. J. Pharm. 1989, 55, 17-23.
    • (1989) Int. J. Pharm. , vol.55 , pp. 17-23
    • Catz, P.1    Friend, R.D.2
  • 25
    • 0034019883 scopus 로고    scopus 로고
    • Microdialysis sampling coupled to HPLC for transdermal delivery study of ondansetron hydrochloride in rats
    • Ding, P.T.; Xu, H.; Wei, G.; Zheng, J.M. Microdialysis sampling coupled to HPLC for transdermal delivery study of ondansetron hydrochloride in rats. Biomed. Chromatogr. 2000, 14, 141-143.
    • (2000) Biomed. Chromatogr. , vol.14 , pp. 141-143
    • Ding, P.T.1    Xu, H.2    Wei, G.3    Zheng, J.M.4
  • 26
    • 0037038304 scopus 로고    scopus 로고
    • In vitro iontophoresis of R-apomorphine across human stratum corneum-structure-transport relationship of penetration enhancement
    • Li, G.L.; Van-der-Geest, R.; Chanet, L.; Van-Zanten, E.; Danhof, M.; Bouwstra, J.A. In vitro iontophoresis of R-apomorphine across human stratum corneum-structure-transport relationship of penetration enhancement. J. Control. Release 2002, 84, 49-57.
    • (2002) J. Control. Release , vol.84 , pp. 49-57
    • Li, G.L.1    Van-Der-Geest, R.2    Chanet, L.3    Van-Zanten, E.4    Danhof, M.5    Bouwstra, J.A.6
  • 27
    • 0035998950 scopus 로고    scopus 로고
    • Terpenes in propylene glycol as skin-penetration enhancers: Permeation and partition of haloperidol, fourier transform infrared spectroscopy, and differential scanning calorimetry
    • Vaddi, H.K.; Ho, P.C.; Chan, S.Y. Terpenes in propylene glycol as skin-penetration enhancers: permeation and partition of haloperidol, fourier transform infrared spectroscopy, and differential scanning calorimetry. J. Pharm. Sci. 2002, 91, 1639-1651.
    • (2002) J. Pharm. Sci. , vol.91 , pp. 1639-1651
    • Vaddi, H.K.1    Ho, P.C.2    Chan, S.Y.3
  • 28
    • 0034868017 scopus 로고    scopus 로고
    • A new colorimetric assay for studying and rapid screening of membrane penetration enhancers
    • Evard, D.; Touitou, E.; Kolusheva, S.; Fishov, Y.; Jelinek, R. A new colorimetric assay for studying and rapid screening of membrane penetration enhancers. Pharm. Res. 2001, 18, 943-949.
    • (2001) Pharm. Res. , vol.18 , pp. 943-949
    • Evard, D.1    Touitou, E.2    Kolusheva, S.3    Fishov, Y.4    Jelinek, R.5
  • 29
    • 0026546284 scopus 로고
    • Propylene glycol as a vehicle for percutaneous absorption of therapeutic agents
    • Bailey, D.N. Propylene glycol as a vehicle for percutaneous absorption of therapeutic agents. J. Anal. Toxicol. 1992, 16, 97-98.
    • (1992) J. Anal. Toxicol. , vol.16 , pp. 97-98
    • Bailey, D.N.1
  • 30
    • 0032934877 scopus 로고    scopus 로고
    • Effect of linolenic acid ethanol or limonene ethanol and iontophoresis on the in vitro percutaneous absorption of LHRH and ultrastructure of human epidermis
    • Bhatia, K.S.; Singh, J. Effect of linolenic acid ethanol or limonene ethanol and iontophoresis on the in vitro percutaneous absorption of LHRH and ultrastructure of human epidermis. Int. J. Pharm. 1999, 180, 235-250.
    • (1999) Int. J. Pharm. , vol.180 , pp. 235-250
    • Bhatia, K.S.1    Singh, J.2
  • 31
    • 0026621780 scopus 로고
    • Enhancement effects in the permeation of alprazolam through hairless mouse skin
    • Carelli, V.; Di Colo, G.; Nannipieri, E.; Serafini, M.F. Enhancement effects in the permeation of alprazolam through hairless mouse skin. Int. J. Pharm. 1992, 88, 89-97.
    • (1992) Int. J. Pharm. , vol.88 , pp. 89-97
    • Carelli, V.1    Di Colo, G.2    Nannipieri, E.3    Serafini, M.F.4
  • 32
    • 0032531673 scopus 로고    scopus 로고
    • Improving insulin enteral absorption using water-in-oil-in-water emulsion
    • Morishita, M.; Matsuzawa, A.; Takayama, K.; Isowa, K.; Nagai, T. Improving insulin enteral absorption using water-in-oil-in-water emulsion. Int. J. Pharm. 1998, 172, 189-198.
    • (1998) Int. J. Pharm. , vol.172 , pp. 189-198
    • Morishita, M.1    Matsuzawa, A.2    Takayama, K.3    Isowa, K.4    Nagai, T.5
  • 33
    • 0037423771 scopus 로고    scopus 로고
    • Transdermal iontophoresis of insulin. V. Effects of terpenes
    • Pillai, O.; Panchagnula, R. Transdermal iontophoresis of insulin. V. Effects of terpenes. J. Control. Release 2003, 88, 287-296.
    • (2003) J. Control. Release , vol.88 , pp. 287-296
    • Pillai, O.1    Panchagnula, R.2
  • 34
    • 0028830178 scopus 로고
    • Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time; permeation, partitioning and differential scanning calorimetry
    • Yamane, M.A.; William, A.C.; Barry, B.W. Effects of terpenes and oleic acid as skin penetration enhancers towards 5-fluorouracil as assessed with time; permeation, partitioning and differential scanning calorimetry. Int. J. Pharm. 1995, 116, 237-251.
    • (1995) Int. J. Pharm. , vol.116 , pp. 237-251
    • Yamane, M.A.1    William, A.C.2    Barry, B.W.3
  • 35
    • 0030787333 scopus 로고    scopus 로고
    • Mechanism of transdermal transport of 5-fluorouracil by terpenes: Carvone, 1,8-cineole and thymol
    • Gao, S.; Singh, J. Mechanism of transdermal transport of 5-fluorouracil by terpenes: carvone, 1,8-cineole and thymol. Int. J. Pharm. 1997, 154, 67-77.
    • (1997) Int. J. Pharm. , vol.154 , pp. 67-77
    • Gao, S.1    Singh, J.2
  • 37
    • 0002054172 scopus 로고    scopus 로고
    • Facilitated transdermal delivery by iontophoresis
    • Bronaugh, R.L., Maibach, H.I., Eds.; Marcel Dekker: New York
    • Singh, P.; Liu, P.; Dinh, S.M. Facilitated transdermal delivery by iontophoresis. In Percutaneous Absorption; Bronaugh, R.L., Maibach, H.I., Eds.; Marcel Dekker: New York, 1999; 633-657
    • (1999) Percutaneous Absorption , pp. 633-657
    • Singh, P.1    Liu, P.2    Dinh, S.M.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.