Mechanism(s) of in vitro percutaneous absorption enhancement of tamoxifen by enhancers

Journal of Pharmaceutical Sciences

Volumn 89, Issue 6, 2000, Pages 771-780

  Zhao, Kaidi ^a   Singh, Jagdish ^a  

^a NORTH DAKOTA STATE UNIVERSITY   (United States)

Author keywords

Enhancers; FT IR; Percutaneous absorption; Tamoxifen; TEWL

Indexed keywords

EUGENOL; LIMONENE; MENTHONE; PROPYLENE GLYCOL; TAMOXIFEN; TERPENE DERIVATIVE;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG BINDING; DRUG DIFFUSION; DRUG PENETRATION; EPIDERMIS; NONHUMAN; PARTITION COEFFICIENT; SKIN ABSORPTION; SKIN WATER LOSS; STRATUM CORNEUM;

EID: 0033812031     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1520-6017(200006)89:6<771::AID-JPS9>3.0.CO;2-Y     Document Type: Article

References (28)

1. Percutaneous absorption of 2', 3'-dideoxyinosine in rats
2. Comparative analysis of percutaneous absorption enhancement by d-limonene and oleic acid based on a skin diffusion model
3. Mechanism of transdermal transport of 5-fluorouracil by terpenes: Carvone, 1,8-cineole, and thymol
4. Terpenes as percutaneous absorption promoter
5. Terpenes penetration enhancers in propylene glycol/water cosolvent systems: Effectiveness and mechanism of action
6. Azone® induced fluidity in human stratum corneum. A Fourier transform infrared spectroscopy investigation using the perdeuterated analogue
7. Enhanced permeation of polar compounds through human epidermis. I. Permeability and membrane structural change in the presence of short-chain alcohols
8. Polymeric phase behavior of phospholipid membranes studied by infrared spectroscopy
9. Enhancing effect of pyrrolidone derivatives on transdermal of 5-fluorouracil, triamcinolone acetonide, indomethacin, and flurbiproben
10. Effect of organic solvents on in vitro human skin water barrier function
11. In vivo relationship between transepidermal water loss and percutaneous penetration of some organic compounds in man: Effect of anatomic site
12. In vivo relationship between percutaneous absorption and transepidermal water loss
13. Endocrine pharmacology of antiestrogens as antitumor agents
14. Effect of penetration enhancers and iontophoresis on the ultrastructure and cholecystokinin-8 permeability through porcine skin
15. Effect of linglenic acid/ethanol or limonene/ethanol and iontophoresis on the in vitro percutaneous absorption of LHRH and ultrastructure of human epidermis
16. Pig ear skin as an in vitro model for human skin permeability
17. Pig ear skin as a model for predicting percutaneous absorption in man
18. In vivo percutaneous absorption of cadium from water and soil into human skin
19. In vitro percutaneous absorption enhancement of a lipophilic drug tamoxifen by terpenes
20. Glyphosate skin binding, absorption, residual tissue distribution, and skin decontamination
21. Structure-activity relationship of 1-alkyl- or 1-alkenyl-azacycloalkanone derivatives as percutaneous penetration enhancers
22. Correction of perfusate concentration for sample removal
23. Examination of the effect of ethanol on human corneum in vivo using infrared spectroscopy
24. Mechanism of transport enhancement of LHRH through porcine epidermis by terpenes and iontophoresis: Permeability and lipid extraction studies
25. Skin permeation enhancement reversibility
26. Effects of surfactants and solvents on the permeability of epidermis