Chemistry and biology of mercaptoacetamides as novel histone deacetylase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 5, 2005, Pages 1389-1392

  Chen, Bin ^a   Petukhov, Pavel A ^a   Jung, Mira ^b   Velena, Alfredo ^b   Eliseeva, Elena ^b   Dritschilo, Anatoly ^b   Kozikowski, Alan P ^a  

^a UNIVERSITY OF ILLINOIS AT CHICAGO   (United States)

^b GEORGETOWN UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

HDAC; Histone deacetylase inhibitor; Mercaptoacetamide

Indexed keywords

ACETAMIDE DERIVATIVE; HISTONE DEACETYLASE INHIBITOR;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER GROWTH; CANCER INHIBITION; DRUG DESIGN; DRUG SYNTHESIS; ENZYME INHIBITION; INHIBITION KINETICS;

EID: 13944274825     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.01.006     Document Type: Article

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