The design and synthesis of novel 3-[2-indol-1-yl-ethyl]-1H-indole derivatives as selective inhibitors of CDK4

Tetrahedron Letters

Volumn 46, Issue 9, 2005, Pages 1423-1425

  Aubry, Carine ^a   Patel, Asma ^a   Mahale, Sachin ^b   Chaudhuri, Bhabatosh ^b   Maréchal, Jean Didier ^a   Sutcliffe, Michael J ^a   Jenkins, Paul R ^a  

^a UNIVERSITY OF LEICESTER   (United Kingdom)

^b DE MONTFORT UNIVERSITY   (United Kingdom)

Author keywords

3 2 Indol 1 yl ethyl 1H indole; CDK4; Fascaplysin; IC50; Indole; Molecular modelling

Indexed keywords

3 (2 INDOL 1 YLETHYL) 1H INDOLE; CYCLIN DEPENDENT KINASE 4; CYCLIN DEPENDENT KINASE INHIBITOR; FASCAPLYSIN; INDOLE DERIVATIVE; INDOLYLETHYLINDOLE; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGICAL ACTIVITY; DRUG DESIGN; DRUG SYNTHESIS;

EID: 13444291631     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2005.01.054     Document Type: Article

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