Crystallographic analysis of potent and selective factor Xa inhibitors complexed to bovine trypsin

Acta Crystallographica Section D: Biological Crystallography

Volumn 55, Issue 8, 1999, Pages 1395-1404

  Whitlow, Marc ^a   Arnaiz, Damain O ^a   Buckman, Brad O ^a   Davey, David D ^a   Griedel, Brain ^a   Guilford, William J ^a   Koovakkat, Sunil K ^a   Liang, Amy ^a   Mohan, Raju ^a   Phillips, Gary B ^a   Seto, Marian ^a   Shaw, Kenneth J ^a   Xu, Wei ^a   Zhao, Zuchun ^a   Light, David R ^a   Morrissey, Michael M ^a  

^a BAYER AG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BLOOD CLOTTING FACTOR 10A; TRYPSIN;

ANIMAL; ARTICLE; CATTLE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; DRUG ANTAGONISM; DRUG DESIGN; ELECTROCHEMISTRY; HUMAN; IN VITRO STUDY; MACROMOLECULE; PROTEIN BINDING; PROTEIN CONFORMATION; X RAY CRYSTALLOGRAPHY;

ANIMALS; CATTLE; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; ELECTROCHEMISTRY; FACTOR XA; HUMANS; MACROMOLECULAR SUBSTANCES; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PROTEIN BINDING; PROTEIN CONFORMATION; TRYPSIN;

EID: 13044286035     PISSN: 09074449     EISSN: None     Source Type: Journal    
DOI: 10.1107/S0907444999007350     Document Type: Article

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