Allostery and cooperativity in the interaction of drugs with ionic channel receptors

Physiological Research

Volumn 53, Issue 6, 2004, Pages 569-579

  Krusek J ^a  

^a INSTITUTE OF PHYSIOLOGY   (Czech Republic)

Author keywords

Affinity; Allostery; Cooperativity; Efficacy; Hill coefficient; Nicotinic acetylcholine receptor

Indexed keywords

ION CHANNEL; NICOTINIC RECEPTOR; RECEPTOR SUBUNIT;

ALLOSTERISM; ANALYTIC METHOD; BINDING SITE; COMPLEX FORMATION; CONFORMATIONAL TRANSITION; COOPERATION; DRUG EFFICACY; DRUG INTERACTION; DRUG RECEPTOR BINDING; NONHUMAN; RECEPTOR UPREGULATION; SHORT SURVEY; THERMODYNAMICS;

ANIMALS; BINDING SITES; HUMANS; ION CHANNEL GATING; ION CHANNELS; KINETICS; MODELS, BIOLOGICAL; MODELS, CHEMICAL; PHARMACEUTICAL PREPARATIONS; PROTEIN BINDING; RECEPTORS, CELL SURFACE;

EID: 11244316778     PISSN: 08628408     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Short Survey

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