Pyrazino[1,2-a]indoles as novel high-affinity and selective imidazoline I2 receptor ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 4, 2004, Pages 1003-1005

  Chang Fong, Jean ^a   Tyacke, Robin J ^b   Lau, Alice ^b   Westaway, Julie ^b   Hudson, Alan L ^b   Glennon, Richard A ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

^b UNIVERSITY OF BRISTOL   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

8 METHOXY 1,2,3,4 TETRAHYDROPYRAZINO[1,2 A]INDOLE; ALPHA 2 ADRENERGIC RECEPTOR; IMIDAZOLINE I1 RECEPTOR; IMIDAZOLINE I2 RECEPTOR; INDOLE DERIVATIVE; PYRAZINO[1,2 A]INDOLE DERIVATIVE; SEROTONIN 2A RECEPTOR; SEROTONIN 2C RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; DRUG SELECTIVITY;

EID: 0842265943     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.12.033     Document Type: Article

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