[3H]2-(2-benzofuranyl)-2-imidazoline: A new selective high affinity radioligand for the study of rabbit brain imidazoline I2 receptors

European Journal of Pharmacology

Volumn 304, Issue 1-3, 1996, Pages 221-229

  Lione, Lisa A ^a   Nutt, David J ^a   Hudson, Alan L ^a  

^a UNIVERSITY OF BRISTOL   (United Kingdom)

Author keywords

clonidine; idazoxan; imidazoline I2 receptor; 3H 2 (2 benzofuranyl) 2 imidazoline

Indexed keywords

2 (2 BENZOFURANYL) 2 IMIDAZOLINE; AGMATINE; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMILORIDE; BACLOFEN; BICUCULLINE; CIRAZOLINE; CLONIDINE; CLORGYLINE; EFAROXAN; GUANABENZ; IDAZOXAN; IMIDAZOLINE DERIVATIVE; IMIDAZOLINE RECEPTOR; MONOAMINE OXIDASE A INHIBITOR; MOXONIDINE; N METHYL DEXTRO ASPARTIC ACID; NAPHAZOLINE; PARGYLINE; PROPRANOLOL; RADIOLIGAND; RAUWOLSCINE; RECEPTOR SUBTYPE; SCOPOLAMINE; SELEGILINE; UNCLASSIFIED DRUG; UNINDEXED DRUG; 2-(2-BENZOFURANYL)-2-IMIDAZOLINE; BENZOFURAN DERIVATIVE; DRUG RECEPTOR; IMIDAZOLE DERIVATIVE; IMIDAZOLINE RECEPTORS;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING COMPETITION; BINDING KINETICS; BINDING SITE; BRAIN MEMBRANE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SELECTIVITY; FEMALE; MALE; NONHUMAN; PRIORITY JOURNAL; RABBIT; RECEPTOR BINDING; AFFINITY LABELING; ANIMAL; BRAIN; CELL MEMBRANE; DRUG ANTAGONISM; IN VITRO STUDY; KINETICS; METABOLISM; PROTEIN BINDING; RADIOASSAY; ULTRASTRUCTURE;

AFFINITY LABELS; ANIMALS; BENZOFURANS; BINDING, COMPETITIVE; BRAIN; CELL MEMBRANE; FEMALE; IMIDAZOLES; KINETICS; MALE; PROTEIN BINDING; RABBITS; RADIOLIGAND ASSAY; RECEPTORS, DRUG;

EID: 0030598574     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00131-8     Document Type: Article

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