An expeditious multigram preparation of the marine protein kinase inhibitor debromohymenialdisine

Tetrahedron Letters

Volumn 44, Issue 52, 2003, Pages 9263-9265

  Portevin, Bernard ^a   Golsteyn, Roy M ^b   Pierré, Alain ^b   De Nanteuil, Guillaume ^a  

^a INSTITUT DE RECHERCHES SERVIER   (France)

^b INSTITUT DE RECHERCHES SERVIER   (France)

Author keywords

Chk1; Debromohymenialdisine

Indexed keywords

DEBROMOHYMENIALDISINE; PROTEIN KINASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; BROMINATION; CYCLIZATION; OXIDATION;

EID: 0344441316     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2003.10.074     Document Type: Article

References (10)

1. Curman D., Cinel B., Williams D.E., Rundle N., Block W.D., Goodarzi A.A., Hutchins J.R., Clarke P.R., Zhou B.-B., Lees-Miller S.P., Andersen R.J., Roberge M. J. Biol. Chem. 276:2001;17914-17919.
2. Tasdemir D., Mallon R., Greenstein M., Feldberg L.R., Kim S.C., Collins K., Wojciechowicz D., Mangalindan G.C., Concepcion G.P., Harper M.K., Ireland C.M. J. Med. Chem. 45:2002;529-532.
3. Meijer L., Thunissen A.M., White A.W., Garnier M., Nikolic M., Tsai L.H., Walter J., Cleverley K.E., Salinas P.C., Wu Y.Z., Mandelkow E.M., Kim S.H., Pettit G.R. Chem. Biol. 7:2000;51-63.
4. Annoura H., Tatsuoka T. Tetrahedron Lett. 36:1995;413-416.
5. Xu Y., Yakushijin K., Horne D.A. J. Org. Chem. 62:1997;456-464.
6. Barrios Sosa A.C., Yakushijin K., Horne D.A. J. Org. Chem. 65:2000;610-611.
7. Prager R.H., Tsopelas C. Aust. J. Chem. 45:1992;1771-1777.
8. Cho H., Matsuki S., Mizuno A., Annoura H., Tatsuoka T. J. Heterocycl. Chem. 34:1997;87-91.
9. Niigata, K.; Okada, M.; Yoneda, T. Australian patent 1987, AU-A-67401/87, 138-9.
10. Lindel T., Hoffmann H. Tetrahedron Lett. 38:1997;8935-8938.