Screening of Plasmodium falciparum iron superoxide dismutase inhibitors and accuracy of the SOD-assays

Bioorganic and Medicinal Chemistry

Volumn 11, Issue 23, 2003, Pages 4941-4944

  Soulère, Laurent ^a,d   Delplace, Patrick ^b   Davioud Charvet, Elisabeth ^c,e   Py, Sandrine ^c,f   Sergheraert, Christian ^c   Périé, Jacques ^a   Ricard, Isabelle ^b   Hoffmann, Pascal ^a   Dive, Daniel ^b  

^a CNRS   (France)

^b INSTITUT PASTEUR DE LILLE   (France)

^c INSTITUT DE BIOLOGIE DE LILLE   (France)

^d MAX PLANCK INSTITUTE OF MOLECULAR PHYSIOLOGY   (Germany)

^e UNIVERSITY OF HEIDELBERG   (Germany)

^f UNIVERSITÉ JOSEPH FOURIER   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AB 93; ANTIMALARIAL AGENT; BB 24; BB 29; BB 31; BB 82; CHLOROQUINE; DS 88; ENZYME INHIBITOR; F 12; IRON; RECOMBINANT ENZYME; SG 5281; SG 7861; SP 112; SP 13; SP 35; SP 59; SP 72; SP 81; SUPEROXIDE DISMUTASE; UNCLASSIFIED DRUG;

ARTICLE; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; DRUG TARGETING; ENZYME ASSAY; NONHUMAN; PLASMODIUM FALCIPARUM;

PLASMODIUM FALCIPARUM;

EID: 0242361212     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2003.09.011     Document Type: Article

References (18)

1. Fridovich I. Annu. Rev. Biochem. 64:1995;97.
2. Parker M.W., Blake C.C. FEBS Lett. 229:1988;377 Jackson S.M., Cooper J.B. Biometals. 11:1998;159.
3. Parker M.W., Blake C.C. FEBS Lett. 229:1988;377 Jackson S.M., Cooper J.B. Biometals. 11:1998;159.
4. Meshnick S.R., Kitchener K.R., Le Trang N. Biochem. Pharmacol. 34:1985;3147.
5. Tabor S., Richardson C.C. Proc. Natl. Acad. Sci. U.S.A. 82:1985;1074.
6. Gratepanche S., Menage S., Touati D., Wintjens R., Delplace P., Fontecave M., Masset A., Camus D., Dive D. Mol. Biochem. Parasitol. 120:2002;237.
7. The synthesis of some of these compounds has previously been published: Salmon-Chemin L., Buisine E., Yardley V., Kohler S., Debreu M.A., Landry V., Sergheraert C., Croft S.L., Krauth-Siegel L.R., Davioud-Charvet E. J. Med. Chem. 44:2001;548 Bonnet B., Soullez D., Girault S., Maes L., Landry V., Davioud-Charvet E., Sergheraert C. Bioorg. Med. Chem. 8:2000;95 Vendeville S., Buisine E., Williard X., Schrevel J., Grellier P., Santana J., Sergheraert C. Chem. Pharm. Bull. 47:1999;194.
8. The synthesis of some of these compounds has previously been published: Salmon-Chemin L., Buisine E., Yardley V., Kohler S., Debreu M.A., Landry V., Sergheraert C., Croft S.L., Krauth-Siegel L.R., Davioud-Charvet E. J. Med. Chem. 44:2001;548 Bonnet B., Soullez D., Girault S., Maes L., Landry V., Davioud-Charvet E., Sergheraert C. Bioorg. Med. Chem. 8:2000;95 Vendeville S., Buisine E., Williard X., Schrevel J., Grellier P., Santana J., Sergheraert C. Chem. Pharm. Bull. 47:1999;194.
9. The synthesis of some of these compounds has previously been published: Salmon-Chemin L., Buisine E., Yardley V., Kohler S., Debreu M.A., Landry V., Sergheraert C., Croft S.L., Krauth-Siegel L.R., Davioud-Charvet E. J. Med. Chem. 44:2001;548 Bonnet B., Soullez D., Girault S., Maes L., Landry V., Davioud-Charvet E., Sergheraert C. Bioorg. Med. Chem. 8:2000;95 Vendeville S., Buisine E., Williard X., Schrevel J., Grellier P., Santana J., Sergheraert C. Chem. Pharm. Bull. 47:1999;194.
10. Ewing J.F., Janero D.R. Anal. Biochem. 232:1995;243.
11. Marklund S., Marklund G. Eur. J. Biochem. 47:1974;469.
12. Desjardins R.E., Canfield C.J., Haynes J.D., Chulay J.D. Antimicrob. Agents Chemother. 16:1979;710.
13. Sines J., Allison S., Wierzbicki A., McCammon J.A. J. Phys. Chem. 94:1990;959.
14. Florent I., Mouray E., Dali Ali F., Drobecq H., Girault S., Schrevel J., Sergheraert C., Grellier P. FEBS Lett. 484:2000;246.
15. Nielsen S.F., Christensen S.B., Cruciani G., Kharazmi A., Liljefors T. J. Med. Chem. 41:1998;4819.
16. Troeberg L., Chen X., Flaherty T.M., Morty R.E., Cheng M., Hua H., Springer C., McKerrow J.H., Kenyon G.L., Lonsdale-Eccles J.D., Coetzer T.H., Cohen F.E. Mol. Med. 6:2000;660.
17. Ram V.J., Saxena A.S., Srivastava S., Chandra S. Bioorg. Med. Chem. Lett. 10:2000;2159.
18. Unpublished result by R. C. Garratt, R. C. (manuscript in preparation).