Identification of inhibitors of an 80 kDa protease from Trypanosoma cruzi through the screening of a combinatorial peptide library

Chemical and Pharmaceutical Bulletin

Volumn 47, Issue 2, 1999, Pages 194-198

  Vendeville, Sandrine ^a   Buisine, Eric ^a   Williard, Xavier ^a   Schrevel, Joseph ^b   Grellier, Philippe ^b   Santana, Jaime ^c   Sergheraert, Christian ^a  

^a CNRS   (France)

^b MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

^c UNIVERSITY OF BRASILIA   (Brazil)

Author keywords

Chagas disease; Combinatorial chemistry; Protease inhibitor; Tetrahydroisoquinoleic acid; Tripeptide; Trypanosoma cruzi

Indexed keywords

ENZYME INHIBITOR; PROTEINASE INHIBITOR; SUAM 1221; TRIPEPTIDE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; ENZYME INHIBITION; NONHUMAN; PEPTIDE ANALYSIS; PROTEIN STRUCTURE; TRYPANOSOMA CRUZI;

EID: 0032941330     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.47.194     Document Type: Article

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