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note
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Ethoxyacetylene was purchased from Lancaster Chemical Co. as an approximately 50%w/w solution in hexanes. Yields 7a-1 were calculated based upon the amount of acid chloride used.
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9a and 9b were prepared in 99% and 92% yields, respectively
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A modification of the method reported in: Newman, M. S.; Geib, J. R.; Stalick, W. M. Org. Prep. Proced. Int. 1972, 4, 89.
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0141661694
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note
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Contrastingly, the reaction of 4 with cyclopenta-1,3-dione required several days for completion under these conditions.
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1-Methyltetrazole-5-sulfenyl chloride has been previously prepared by chlorination of the mercaptan with chlorine. See: Postle, S. R. U.S. Patent 4 387 158, 1983.
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Postle, S.R.1
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