N-(3-Phenylsulfonyl-3-piperidinoyl)-phenylalanine derivatives as potent, selective VLA-4 antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 5, 2003, Pages 885-890

  Gutteridge, Clare E ^a,b   De Laszlo, Stephen E ^a   Kamenecka, Theodore M ^a   McCauley, Ermengilda ^a   Van Riper, Gail ^a   Mumford, Richard A ^a   Kidambi, Usha ^a   Egger, Linda A ^a   Tong, Sharon ^a   Hagmann, William K ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

^b UNITED STATES NAVAL ACADEMY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 SULFONYLCYCLOPENTYL CARBOXYLIC ACID AMIDE; AMIDE; BETA1 INTEGRIN; INTEGRIN; LIGAND; N (3 PHENYLSULFONYL 3 PIPERIDINOYL) 4 (2',6' DIMETHOXYPHENYL)PHENYLALANINE; N (3 PHENYLSULFONYL 3 PIPERIDINOYL)PHENYLALANINE DERIVATIVE; PHENYLALANINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; STRUCTURE ACTIVITY RELATION;

EID: 0037430555     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)01077-6     Document Type: Article

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