Integrastatins: Structure and HIV-1 integrase inhibitory activities of two novel racemic tetracyclic aromatic heterocycles produced by two fungal species

Tetrahedron Letters

Volumn 43, Issue 13, 2002, Pages 2351-2354

  Singh, Sheo B ^a   Zink, Deborah L ^a   Quamina, Donette S ^a   Pelaez, Fernando ^b   Teran, Ana ^b   Felock, Peter ^a   Hazuda, Daria J ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

^b Medical affairs Merck sharp and Dohme ltd   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; AROMATIC COMPOUND; HETEROCYCLIC COMPOUND; INTEGRASE; INTEGRASE INHIBITOR; INTEGRASTIN A; INTEGRASTIN B; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG STRUCTURE; ENZYME INHIBITION; FERMENTATION; FUNGUS; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; MASS SPECTROMETRY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; RACEMIC MIXTURE;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0037170622     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(02)00265-4     Document Type: Article

References (10)