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Journal of the American Chemical Society

Volumn 124, Issue 2, 2002, Pages 205-215

Calorimetric and structural studies of 1,2,3-trisubstituted cyclopropanes as conformationally constrained peptide inhibitors of Src SH2 domain binding

(5) Davidson, James P a Lubman, Olga b Rose, Thierry b Waksman, Gabriel b Martin, Stephen F a

a UNIVERSITY OF TEXAS AT AUSTIN (United States)

b WASHINGTON UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ISOTHERMAL TITRATION CALORIMETRY;

COMPLEXATION; CRYSTAL STRUCTURE; ENZYMES; STRUCTURE (COMPOSITION); THERMODYNAMIC PROPERTIES; X RAY CRYSTALLOGRAPHY;

PROPANE;

CYCLOPROPANE DERIVATIVE; LIGAND; OLIGOPEPTIDE; PHOSPHOTYROSINE; PHOSPHOTYROSYLGLUTAMYLGLUTAMYLISOLEUCINE; PROTEIN KINASE INHIBITOR; PROTEIN KINASE P60; TETRAPEPTIDE; TYROSINE; UNCLASSIFIED DRUG;

ARTICLE; CALORIMETRY; COMPLEX FORMATION; CRYSTAL STRUCTURE; ENTHALPY; ENTROPY; ENZYME BINDING; ENZYME CONFORMATION; ENZYME INHIBITOR INTERACTION; PROTEIN QUATERNARY STRUCTURE; STEREOSPECIFICITY; STRUCTURE ANALYSIS; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CALORIMETRY; CRYSTALLOGRAPHY, X-RAY; CYCLOPROPANES; ENZYME INHIBITORS; MOLECULAR MIMICRY; OLIGOPEPTIDES; PHOSPHOPEPTIDES; PHOSPHOTYROSINE; PROTEIN CONFORMATION; PROTEIN STRUCTURE, TERTIARY; SRC HOMOLOGY DOMAINS; SRC-FAMILY KINASES; STRUCTURE-ACTIVITY RELATIONSHIP; THERMODYNAMICS;

EID: 0037116524 PISSN: 00027863 EISSN: None Source Type: Journal
DOI: 10.1021/ja011746f Document Type: Article

Times cited : (84)

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